首页> 外文期刊>Acta Pharmacologica Sinica >Protection of dopaminergic antagonists against anoxia-induced inhibition of Ca~2+ -calmodulin dependent protein kinase Ⅱ activity in rat brain
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Protection of dopaminergic antagonists against anoxia-induced inhibition of Ca~2+ -calmodulin dependent protein kinase Ⅱ activity in rat brain

机译:多巴胺能拮抗剂对缺氧诱导的大鼠脑Ca〜2 +-钙调蛋白依赖性蛋白激酶Ⅱ活性的抑制作用

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摘要

AIM: To study the effect of dopamine receptor antagonists on anoxia-induced inhibition of Ca~2+ - calmodulin dependent protein kinase Ⅱ (CCDPK Ⅱ) activity in rat hippocampus and striatum. METHODS: Using the rat hippocampal and striatal Slices under 95 /100 N_2 + 5 /100 CO_2, the activity of CCDPK Ⅱ was examined by ~32P-incorporation. CONCLUSION: Dopamine receptor stimulation is involved in anoxia- Induced inhibition of CCDPK Ⅱ activity in rat Hippocampus and striatum.
机译:目的:研究多巴胺受体拮抗剂对缺氧诱导的大鼠海马和纹状体Ca〜2 +-钙调蛋白依赖性蛋白激酶Ⅱ(CCDPKⅡ)活性的抑制作用。方法:在95/100 N_2 + 5/100 CO_2下的海马和纹状体切片,通过〜32P掺入法检测CCDPKⅡ的活性。结论:多巴胺受体刺激参与了缺氧诱导的大鼠海马和纹状体对CCDPKⅡ活性的抑制。

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