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机译:Structure activity study of S-trityl-cysteamine dimethylaminopyridine derivatives as SIRT2 inhibitors: Improvement of SIRT2 binding and inhibition
Sci Farm Ltd, Dept Drug Discovery, Chuo Ku, 1-7-30-80-5 Kuhonji, Kumamoto 8620976, Japan;
Kumamoto Univ, Fac Life Sci, Med & Biol Chem Sci Farm Joint Res Lab, Chuo Ku, 5-1 Oe Honmachi;
RIKEN, Seed Cpds Exploratory Unit Drug Discovery Platfor, Ctr Sustainable Resource Sci, 2-1RIKEN, Chem Genom Res Grp, Ctr Sustainable Resource Sci, 2-1 Hirosawa, Wako, Saitama 3510198, Japan;
SIRT2; S-trityl-L-cysteine; S-trityl cysteamine; Molecular docking; Selectivity pocket;