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机译:Structure-based discovery of selective positive allosteric modulators of antagonists for the M-2 muscarinic acetylcholine receptor
Monash Univ, Monash Inst Pharmaceut Sci, Drug Discovery Biol, Parkville, Vic 3052, Australia;
Univ Calif San Francisco, Dept Pharmaceut Chem, San Francisco, CA 94158 USA;
Univ Calif San Diego, Sch Med, Dept Pharmacol, La Jolla, CA 92093 USATsinghua Univ, Sch Med, Beijing Adv Innovat Ctr Struct Biol, Beijing 100084, Peoples R ChinaStanford Univ, Sch Med, Dept Mol & Cellular Physiol, Stanford, CA 94305 USAHarvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA;
GPCR; subtype selectivity; PAM antagonist; docking; structure-based ligand discovery;