首页> 外国专利> METHOD FOR MANUFACTURING FORMULATION CONTAINING SITAGLIPTIN IMMEDIATE RELEASE LAYER, FORMULATION MANUFACTURED BY METHOD, METHOD FOR COATING SITAGLIPTIN IMMEDIATE RELEASE LAYER, AND COMPOSITION FOR COATING SITAGLIPTIN IMMEDIATE RELEASE LAYER

METHOD FOR MANUFACTURING FORMULATION CONTAINING SITAGLIPTIN IMMEDIATE RELEASE LAYER, FORMULATION MANUFACTURED BY METHOD, METHOD FOR COATING SITAGLIPTIN IMMEDIATE RELEASE LAYER, AND COMPOSITION FOR COATING SITAGLIPTIN IMMEDIATE RELEASE LAYER

机译:制造包含西格列汀立即释放层的配方的方法,用该方法制造的制剂,涂覆西格列汀立即释放层的方法以及涂覆西格列汀立即释放层的组合物

摘要

The present invention relates to a method for manufacturing a formulation containing a sitagliptin immediate release layer which comprises following steps of: (a) manufacturing a coating solution by dissolving sitagliptin or pharmaceutically acceptable salt in a highly volatile solvent; and (b) coating a sustained release layer with the coating solution. The present invention also relates to the formulation manufactured by the manufacturing method, a method for coating the sitagliptin immediate release layer, and a composition for coating the sitagliptin immediate release layer. According to the present invention, the coating time can be shortened and the occurrence of a flexible material can be prevented.;COPYRIGHT KIPO 2020
机译:本发明涉及一种包含西他列汀速释层的制剂的制备方法,该方法包括以下步骤:(a)通过将西他列汀或药学上可接受的盐溶解在高挥发性溶剂中来制备包衣溶液; (b)用所述包衣溶液包衣缓释层。本发明还涉及通过该制造方法制造的制剂,涂覆西他列汀速释层的方法和涂覆西他列汀速释层的组合物。根据本发明,可以缩短涂覆时间并且可以防止柔性材料的出现。COPYRIGHT KIPO 2020

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