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Extended release liquid compositions of guanfacine

机译:胍法辛的缓释液体组合物

摘要

The present invention relates to extended release liquid compositions of guanfacine. The extended release liquid compositions of the present invention are bioequivalent to marketed extended release tablet compositions of guanfacine. Said extended release liquid compositions provide substantially similar in-vitro dissolution release profile upon storage for at least seven days. Further, the extended release liquid compositions are stable. The extended release liquid compositions are in the form of ready-to-use liquid compositions or reconstituted liquid compositions. It also relates to processes for the preparation of said extended release liquid compositions.
机译:本发明涉及胍法辛的缓释液体组合物。本发明的缓释液体组合物与市售的胍法辛缓释片剂组合物在生物上等效。所述缓释液体组合物在储存至少七天时提供基本上相似的体外溶出释放曲线。此外,该缓释液体组合物是稳定的。缓释液体组合物为即用型液体组合物或重构的液体组合物的形式。它还涉及用于制备所述缓释液体组合物的方法。

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