首页> 外国专利> 56--4--4H-12-14 4--6H-12-14 NOVEL ANTIFUNGAL 56-DIHYDRO-4-DIFLUOROETHYLPHENYL-4H-PYRROLO12-14BENZODIAZEPINE AND 4-DIFLUOROETHYLPHENYL-6H-PYRROLO12-14BENZODIAZEPINE DERIVATIVES

56--4--4H-12-14 4--6H-12-14 NOVEL ANTIFUNGAL 56-DIHYDRO-4-DIFLUOROETHYLPHENYL-4H-PYRROLO12-14BENZODIAZEPINE AND 4-DIFLUOROETHYLPHENYL-6H-PYRROLO12-14BENZODIAZEPINE DERIVATIVES

机译：56--4-[]-4H- [12-] [14] 4--6H- [12-] [14]新型抗真菌药56-二氢-4- [二氟乙基苯基] -4H-吡咯[12-] [14 ]苯并二氮杂卓和4-二氟乙基苯基-6H-吡咯[12-] [14]苯并二氮杂卓衍生物

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摘要

The present invention relates to novel compounds of formula (I) wherein R ¹ , R ² , R ³ , R ⁴ , R ⁵ and R ⁶ have the meanings as defined in the claims. The compounds according to the present invention are mainly active against dermatophytes and systemic fungal infections. The present invention also relates to a process for the preparation of these novel compounds, pharmaceutical compositions comprising the compounds as active ingredients and their use as medicaments.

机译：本发明涉及式（I）的新型化合物，其中R ^{1 ，R ^{2 ，R ^{3 ，R ^{4 ，R ^{5 和R ^{6 具有权利要求中定义的含义。根据本发明的化合物主要对皮肤真菌和全身性真菌感染具有活性。本发明还涉及这些新型化合物的制备方法，包含该化合物作为活性成分的药物组合物及其作为药物的用途。}}}}}}

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公开/公告号KR101886136B1

专利类型
公开/公告日2018-08-07

原文格式PDF
申请/专利权人 얀센 파마슈티카 엔.브이.;
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申请/专利号KR20127030661
发明设计人 미르포엘 리벤;매스 루이스 줄리스 로게르 마리에;데 비트 켈리;
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申请日2011-06-01
分类号C07D487/04;A61K31/5517;A61P31/10;
国家 KR
入库时间 2022-08-21 12:37:23

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