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METHOD OF IMPROVING COGNITION AND SOCIAL BEHAVIOR IN HUMANS HAVING DEFICITS THEREIN DUE TO NEUROLOGICAL DISORDERS AND COMPOUNDS AND COMPOSITIONS THEREFOR

机译:改善由于神经疾病,化合物及其成分而造成人的认知和社会行为不足的方法

摘要

A β1-ADR agonist prodrug compound, which is hydrolysable in vivo to release a β1-ADR agonist compound, and which prodrug compound contains a group which imparts greater lipophilicity and CNS bioavailability to the prodrug compound relative to the β1-ADR agonist compound.
机译:β1-ADR激动剂前药化合物,其在体内可水解以释放β1-ADR激动剂化合物,并且该前药化合物包含相对于β1-ADR激动剂化合物赋予该前药化合物更大的亲脂性和CNS生物利用度的基团。

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