首页> 外国专利> ARYL-HYDROXYETHYLAMINO-PYRIMIDINES AND TRIAZINES AS MODULATORS OF FATTY ACID AMIDE HYDROLASE

ARYL-HYDROXYETHYLAMINO-PYRIMIDINES AND TRIAZINES AS MODULATORS OF FATTY ACID AMIDE HYDROLASE

机译:芳酰羟乙基氨基嘧啶和三嗪作为脂肪酸酰胺水解酶的调节剂

摘要

Certain aryl-hydroxyethylamino-pyrimidine and triazine compounds aredescribed, which are useful as FAAH inhibitors.Such compounds may be used in pharmaceutical compositions and methods for thetreatment of disease states, disorders,and conditions mediated by fatty acid amide hydrolase (FAAH) activity, such asanxiety, pain, inflammation, sleep disorders,eating disorders, energy metabolism disorders, and movement disorders (e.g.,multiple sclerosis). Methods of synthesizing suchcompounds are also disclosed.
机译:某些芳基-羟乙基氨基-嘧啶和三嗪化合物是所述,其可用作FAAH抑制剂。此类化合物可用于药物组合物和用于治疗疾病,失调,和脂肪酸酰胺水解酶(FAAH)活性介导的条件,例如焦虑,疼痛,炎症,睡眠障碍,饮食失调,能量代谢失调和运动失调(例如,多发性硬化症)。合成这样的方法还公开了化合物。

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