首页> 外国专利> G-RICH ISODNA SEQUENCES FORMING G-QUADRUPLEX STRUCTURE, THEIR FUNCTION AS APTAMERS AND A PROCESS FOR THE PREPARATION THEREOF

G-RICH ISODNA SEQUENCES FORMING G-QUADRUPLEX STRUCTURE, THEIR FUNCTION AS APTAMERS AND A PROCESS FOR THE PREPARATION THEREOF

机译:富含G的ISODNA序列,形成G-四链结构,它们作为适体的功能及其制备方法

摘要

The present invention relates to G-quadruplex forming isoDNA aptamers and a process for the preparation thereof. The present invention further relates to a stable, non-genetic, guanine rich 2'- 5' linked isoDNA selected from 3' deoxy 2'-5' isoDNA and 3' deoxy 2' -5' isoDNA-isoRNA hybrid. The instant 2'-5' linked isoDNA such as the thrombin binding aptamer (isoTBA) can be used in deep vein thrombosis, where prolonged anticoagulant activity is required.
机译:本发明涉及形成G-四链体的isoDNA适体及其制备方法。本发明进一步涉及选自3'脱氧2'-5'异DNA和3'脱氧2'-5'异DNA-isoRNA杂交体的稳定的,非遗传的,富含鸟嘌呤的2'-5'连接的isoDNA。本发明的2'-5'连接的isoDNA,例如凝血酶结合适体(isoTBA)可用于需要延长抗凝活性的深部静脉血栓形成。

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