首页> 外国专利> IDENTIFICATION OF SMALL-MOLECULE CANDIDATE THERAPEUTICS CAPABLE OF INHIBITING OR INTERFERING WITH A TARGET PROTEIN-PROTEIN INTERACTION

IDENTIFICATION OF SMALL-MOLECULE CANDIDATE THERAPEUTICS CAPABLE OF INHIBITING OR INTERFERING WITH A TARGET PROTEIN-PROTEIN INTERACTION

机译:能够抑制或干扰靶蛋白-蛋白相互作用的小分子候选药物的鉴定

摘要

The present invention provides a method of screening method small-molecule candidate therapeutics capable of inhibiting or interfering with intracellular protein-protein interactions, such as cancer associated oncogenic protein interactions and in particular RAS and LMO2 protein-protein interactions. The present invention also provides methods and assays for rationalized drug design based on identifying small molecular weight protein-protein interaction inhibitor molecules that emulate antibody therapeutics products.
机译:本发明提供了一种筛选方法的小分子候选疗法的方法,所述候选疗法能够抑制或干扰细胞内蛋白质-蛋白质相互作用,例如与癌症相关的致癌蛋白质相互作用,特别是RAS和LMO2蛋白质-蛋白质相互作用。本发明还提供了基于鉴定模拟抗体治疗产品的小分子量蛋白质-蛋白质相互作用抑制剂分子的用于合理化药物设计的方法和测定法。

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