首页> 外国专利> Piperidinicos acid Esters Derivatives of biphenyl - 2 - il - carbamic, Muscarinic m3 Receptor Antagonists, Pharmaceutical compositions containing them and Uses Thereof for the treatment of digestive disorders, respiratory and / or urinals.

Piperidinicos acid Esters Derivatives of biphenyl - 2 - il - carbamic, Muscarinic m3 Receptor Antagonists, Pharmaceutical compositions containing them and Uses Thereof for the treatment of digestive disorders, respiratory and / or urinals.

机译：Piperidinicos acid Esters联苯-2-基氨基甲酸的衍生物，毒蕈碱型m3受体拮抗剂，含有它们的药物组合物及其在治疗消化系统疾病，呼吸道和/或小便池中的用途。

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摘要

Claim 1: a compound of formula (1) or pharmaceutically acceptable salts or solvates thereof, or pharmaceutically acceptable salts of said Compounds, in which X is selected: - CH2 - CH2 - C (= o) -, - C (= o) - R1 is H or Methyl; or, alternatively, when X is - CH2 -, then R1 PU DTS also represent a group of Formula 2: in one of R6, R7, R8 and R9 is Oh, one of R6, R7,R8 and R9 is Halo, one of R6, R7, R8 and R9 is H and one of R6, R7, R8 and R9 is selected from H or Halo; one of R2, R3, R4 and R5 is one Oh, R2, R3, R4 and R5 is one of H, R2, R3, R4 and R5 is Halo and one of R2, R3, R4 and R5 is H or Halo or, alternatively, when X is CH2 - C (= o) - R and R1 is Methyl, pue Also be oh, while R2, R3 and R5 are H.

机译：权利要求1：式（1）的化合物或其药学上可接受的盐或溶剂化物，或所述化合物的药学上可接受的盐，其中选择X：-CH 2 -CH 2 -C（＝ o）-，-C（＝ o） -R 1为H或甲基;或者，当X为-CH2-时，R1 PU DTS也代表式2的基团：在R6，R7，R8和R9中的一个为Oh时，R6，R7，R8和R9中的一个为Halo，为一个R6，R7，R8和R9是H，并且R6，R7，R8和R9之一选自H或Halo; R2，R3，R4和R5之一是一个哦，R2，R3，R4和R5是H，R2，R3，R4和R5之一是Halo，而R2，R3，R4和R5之一是H或Halo或，或者，当X为CH2-C（= o）-R并且R1为甲基时，pue也为OH，而R2，R3和R5为H。

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公开/公告号AR072802A1

专利类型
公开/公告日2010-09-22

原文格式PDF
申请/专利权人 PFIZER LIMITED;
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申请/专利号AR2009P102622
发明设计人
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申请日2009-07-13
分类号C07D211/46;A61K31/4465;A61P11/00;A61P11/06;A61P11/08;A61P1/00;A61P13/00;
国家 AR
入库时间 2022-08-21 18:47:29

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