首页> 外国专利> New N-azinyl-N'-pyridylsulfonyl-urea compounds useful e.g. as herbicide, plant growth regulator and plant protection regulator and to combat undesirable plant growth e.g. Agrostis in special plant cultures e.g. wheat, barley and rye

New N-azinyl-N'-pyridylsulfonyl-urea compounds useful e.g. as herbicide, plant growth regulator and plant protection regulator and to combat undesirable plant growth e.g. Agrostis in special plant cultures e.g. wheat, barley and rye

机译:新的N-叠氮基-N'-吡啶基磺酰基-脲化合物可用于例如作为除草剂,植物生长调节剂和植物保护调节剂,并与不希望的植物生长作斗争,例如特殊植物培养中的草小麦,大麦和黑麦

摘要

N-Azinyl-N'-pyridylsulfonyl-urea compounds (I) and their salts are new. N-Azinyl-N'-pyridylsulfonyl-urea compounds of formula (I) and their salts are new. V 1, W 1, X, Y 1N or C (both optionally substituted by R 8); A : N or CR 9; R 9H (preferred), alkyl, halo or haloalkyl; R 1H, alkyl, alkoxy, alkoxyalkyl, alkenyl, alkynyl, cycloalkyl, cycloalkylalkyl, aralkyl or aryl; R 2, R 3alkyl, alkoxy, alkylthio, alkyl amino or dialkylamino (all optionally halo substituted), H or halo; R 4-R 7H, halo, CN, alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, dialkylamino, alkylcarbonyl, alkoxycarbonyl, alkylaminocarbonyl or dialkylaminocarbonyl (where R 4and R6, and/or R 5and R 7is an alkylidene group optionally interrupted by O or S); R 8H, halo, CN, thiocyanato, nitro, alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkyl amino, dialkylamino, alkyl carbonyl, alkoxycarbonyl, alkylaminocarbonyl, or dialkylaminocarbonyl; and Q : O or S. Where one of the residue of V 1, W 1, X, Y 1is N and the remaining residues are C. Independent claims are included for: (1) a (4,5-dihydroisoxazol-3-yl) sulfonamide compound of formula (II); (2) a (4,5-dihydroisoxazol-3-yl) sulfonic acid halide compound of formula (VIII); (3) a (4,5-dihydroisoxazol-3-yl) halide compound of formula (XI); (4) a (4,5-dihydroisoxazol-3-yl) thiol compound of formula (X); and (5) the preparation of (I). Hal : halogen atom. [Image] [Image] [Image] ACTIVITY : Herbicide; Plant Growth Regulant. The herbicidal activity of (I) was tested against Alopecurus myosuroides. The results showed that N-[(4-chloro-6-methoxy-pyrimidin-2-yl)carbamoyl]-3-(4,5-dihydroisoxazol-3-yl)-pyridin-2-sulfonamide exhibited an aborticide effectof 100%. MECHANISM OF ACTION : None given.
机译:N-叠氮基-N'-吡啶基磺酰基-脲化合物(I)及其盐是新的。式(I)的N-叠氮基-N'-吡啶基磺酰基-脲化合物及其盐是新的。 V 1>,W 1>,X,Y 1> N或C(均被R 8任选取代); A:N或CR 9>; R 9> H(优选),烷基,卤素或卤代烷基; R 1> H,烷基,烷氧基,烷氧基烷基,烯基,炔基,环烷基,环烷基烷基,芳烷基或芳基; R 2>,R 3>烷基,烷氧基,烷硫基,烷基氨基或二烷基氨基(全部任选被卤素取代),H或卤素; R 4> -R 7> H,卤素,CN,烷基,烷氧基,烷硫基,烷基亚磺酰基,烷基磺酰基,烷基氨基,二烷基氨基,烷基羰基,烷氧基羰基,烷基氨基羰基或二烷基氨基羰基(其中R 4>和R 6和/或R 5>和R 7>是任选地被O或S中断的亚烷基。 R 8> H,卤素,CN,硫氰酸根,硝基,烷基,烷氧基,烷硫基,烷基亚磺酰基,烷基磺酰基,烷基氨基,二烷基氨基,烷基羰基,烷氧基羰基,烷基氨基羰基或二烷基氨基羰基; V 1>,W 1>,X,Y 1>的残基之一为N且其余残基为C的情况。独立权利要求包括:(1)a(4,5-式(II)的二氢异恶唑-3-基)磺酰胺化合物; (2)式(VIII)的(4,5-二氢异恶唑-3-基)磺酸卤化物; (3)式(XI)的(4,5-二氢异恶唑-3-基)卤化物; (4)式(X)的(4,5-二氢异恶唑-3-基)硫醇化合物; (5)制备(I)。 Hal:卤素原子。 [图片] [图片] [图片]活动:除草剂;植物生长调节剂。测试了(I)的除草剂Aurocurus myosuroides的除草活性。结果表明,N-[(4-氯-6-甲氧基-嘧啶-2-基)氨基甲酰基] -3-(4,5-二氢异恶唑-3-基)-吡啶-2-磺酰胺的杀人效果为100% 。作用机理:未给出。

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