首页> 外国专利> USE OF CETRORELIX FOR THE TREATMENT OF BENIGNA HYPERTROPHY OF PROSTATA AND CANCER DE PROSTATA.

USE OF CETRORELIX FOR THE TREATMENT OF BENIGNA HYPERTROPHY OF PROSTATA AND CANCER DE PROSTATA.

机译:CETRORELIX在前列腺增生和前列腺癌治疗中的应用。

摘要

THE INVENTION REFERS TO A PROCEDURE FOR THE THERAPEUTIC MANAGEMENT OF A BENIGN PROSTATIC HYPERPLASIA AND OF A PROSTATIC CANCER THAT USES CETRORELIX ONLY OR IN COMBINATION WITH THE INHIBITORS OF THE AL-REDUCTAASE OR WITH BLOCKING AGENTS OF THE ALLOCATORS. THE PROCEDURE REDUCES THE VOLUME OF THE PROSTATE AND AVOIDS THE COLLATERAL EFFECTS ASSOCIATED WITH THE TESTOSTERONE LEVELS THAT ARE LOCATED IN THE CASTRATION BAND. CETRORELIX IS ADMINISTERED IN DOSE OF BETWEEN 0.5 MG / DAY AND 20 MG / WEEK OR BETWEEN 0.014 MG / KG BODY WEIGHT PER DAY AND 0.30 MG / KG BODY WEIGHT PER WEEK OR AT LEVELS AROUND BETWEEN 25 AND 125 MG OF CETRORELIX PER MONTH OR BETWEEN 0.376 MG / KG AND 1.71 MG / KG PER MONTH. CETRORELIX CAN BE ADMINISTERED WITH INHIBITORS OF THE -REDUCTASE OR WITH BLOCKING AGENTS OF THE AL-RECEIVERS.
机译:本发明涉及一种对良性前列腺增生症和前列腺癌进行治疗性治疗的方法,该方法仅使用西妥昔单抗或与α-还原酶抑制剂或与分配剂的阻断剂结合使用。该方法减少了前列腺的体积,并避免了与在隔离带中定位的睾丸激素水平相关的结肠影响。 CETRORELIX的剂量介于每天0.5 MG和20 MG /周之间,或每天0.014 MG / KG体重与每周0.30 MG / KG体重之间,或介于每月25到125 MG CETRORELIX之间每月0.376毫克/公斤和1.71毫克/公斤。可以使用-还原酶抑制剂或al受体阻滞剂来抑制CETRORELIX。

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