首页> 外国专利> ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROBENZAZEPINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN.

ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROBENZAZEPINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN.

机译:芳基和异芳基取代的四氢苯并ZE庚因,并用其阻断去甲肾上腺素,多巴胺和血清素的再摄取。

摘要

The compounds of the present invention are represented by the following aryl- and heteroaryl-substituted tetrahydrobenzazepine and dihydrobenzazapine derivatives having formulae I(A-E) and formula (II) where the carbon atom designated * is in the R or S configuration, and the substituents X and Rsup1/sup-Rsup9/sup are as defined herein.
机译:本发明的化合物由以下具有式I(AE)和式(II)的芳基和杂芳基取代的四氢苯并ze庚因和二氢苯并氮杂pine衍生物表示,其中*表示的碳原子为R或S构型,且取代基为X和R 1 -R 9 如本文所定义。

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