as its separate isomers or their mixture, its salt and their hydrates wherein R1 represents cyclic alkyl group comprising 3-6 carbon atoms that can comprise a substitute chosen from halogen atom; R2 represents hydrogen atom; R3 represents hydrogen atom; R4 represents hydrogen atom, amino-group, hydroxyl group; A represents nitrogen atom or part of structure as given in the invention claim; each R5 and R6 represents independently alkyl group comprising 1-6 carbon atoms or hydrogen atom; n means a whole number 1 or 2. Also, invention describes antibacterial agent and therapeutic agent based on compounds of the formula (I) used in treatment of infectious disease, a method for preparing antibacterial agent, a method for preparing a medicinal agent used in treatment of infectious disease and using compound of the formula (I) for preparing an antibacterial agent and using compound of the formula (I) for preparing a medicinal agent used in treatment of infectious disease. Invention provides novel compounds possessing useful biological properties.;EFFECT: improved preparing method of agents, valuable medicinal properties of compounds and agents.;35 cl, 2 tbl, 15 ex"/>
DEHALOGENATED COMPOUNDS, ANTIBACTERIAL AGENT AND THERAPEUTIC AGENT BASED ON THEREOF, METHOD FOR PREPARING ANTIBACTERIAL OR MEDICINAL AGENT, USING DEHALOGENATED COMPOUNDS FOR PREPARING ANTIBACTERIAL OR MEDICINAL AGENT
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DEHALOGENATED COMPOUNDS, ANTIBACTERIAL AGENT AND THERAPEUTIC AGENT BASED ON THEREOF, METHOD FOR PREPARING ANTIBACTERIAL OR MEDICINAL AGENT, USING DEHALOGENATED COMPOUNDS FOR PREPARING ANTIBACTERIAL OR MEDICINAL AGENT
DEHALOGENATED COMPOUNDS, ANTIBACTERIAL AGENT AND THERAPEUTIC AGENT BASED ON THEREOF, METHOD FOR PREPARING ANTIBACTERIAL OR MEDICINAL AGENT, USING DEHALOGENATED COMPOUNDS FOR PREPARING ANTIBACTERIAL OR MEDICINAL AGENT
FIELD: organic chemistry, chemical technology, medicine, pharmacy.;SUBSTANCE: invention relates to a synthetic quinolone agent that is effective as medicinal agents, veterinary preparations, drugs used in fishing industry or as antibacterial preserving agents. Invention describes compound represented by the following general formula (I): as its separate isomers or their mixture, its salt and their hydrates wherein R1 represents cyclic alkyl group comprising 3-6 carbon atoms that can comprise a substitute chosen from halogen atom; R2 represents hydrogen atom; R3 represents hydrogen atom; R4 represents hydrogen atom, amino-group, hydroxyl group; A represents nitrogen atom or part of structure as given in the invention claim; each R5 and R6 represents independently alkyl group comprising 1-6 carbon atoms or hydrogen atom; n means a whole number 1 or 2. Also, invention describes antibacterial agent and therapeutic agent based on compounds of the formula (I) used in treatment of infectious disease, a method for preparing antibacterial agent, a method for preparing a medicinal agent used in treatment of infectious disease and using compound of the formula (I) for preparing an antibacterial agent and using compound of the formula (I) for preparing a medicinal agent used in treatment of infectious disease. Invention provides novel compounds possessing useful biological properties.;EFFECT: improved preparing method of agents, valuable medicinal properties of compounds and agents.;35 cl, 2 tbl, 15 ex
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机译：技术领域本发明涉及一种合成的喹诺酮剂，该喹诺酮剂可有效地用作药物，兽药，用于渔业的药物或用作抗菌防腐剂。本发明描述了由以下通式（I）表示的化合物：<图像文件=“ 00000002.GIF” he =“ 45” id =“ imag00000002” imgContent =“ undefined” imgFormat =“ GIF” wi =“ 86” />如其单独的异构体或它们的混合物，其盐和其水合物，其中R 1 代表包含3-6个碳原子的环烷基，该环烷基可以包含选自卤素原子的取代基; R 2 代表氢原子; R 3 代表氢原子; R 4 代表氢原子，氨基，羟基; A代表本发明权利要求中给出的氮原子或部分结构; R 5 和R 6 分别独立地表示具有1-6个碳原子或氢原子的烷基。 n表示1或2的整数。另外，本发明描述了基于式（I）的化合物的用于治疗传染病的抗菌剂和治疗剂，制备抗菌剂的方法，制备用于细菌的药物的方法。传染性疾病的治疗，并使用式（I）的化合物制备抗菌剂，以及将式（I）的化合物用于制备用于传染病治疗的药物。本发明提供了具有有用的生物学特性的新型化合物。效果：改进了试剂的制备方法，化合物和试剂的有价值的药物特性。35 cl，2 tbl，15 ex
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