首页> 外国专利> VANILLOID ANALOGUES CONTAINING RESINIFERATOXIN PHARMACOPHORES AS POTENT VANILLOID RECEPTOR AGONISTS AND ANALGESICS, COMPOSITIONS AND USES THEREOF

VANILLOID ANALOGUES CONTAINING RESINIFERATOXIN PHARMACOPHORES AS POTENT VANILLOID RECEPTOR AGONISTS AND ANALGESICS, COMPOSITIONS AND USES THEREOF

机译:含有类视紫红质毒素药剂的香草酸类似物,作为强效香草酸受体激动剂和止痛剂,成分和用途

摘要

The present invention is related to new vanilloid analogues containing resiniferatoxin pharmacophores, pharmaceutical compositions comprising such analogues, and their uses as vanilloid receptor agonists and potent analgesics. The present invention provides a pharmaceutical composition for treating acute, chronic, inflammatory or neuropathic pains or for treating bladder hypersensitivity.
机译:本发明涉及含有树脂鞭毛毒素药效基团的新的类香草素类似物,包含此类类似物的药物组合物,以及它们作为类香草素受体激动剂和有效止痛药的用途。本发明提供了用于治疗急性,慢性,炎性或神经性疼痛或用于治疗膀胱超敏反应的药物组合物。

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