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CONCANAMICIN ANALOG, VACUOLAR PROTONE ATP HYDROLASE INHIBITOR, APOTOSIS INDUCER AND ANTICANCER AGENT
CONCANAMICIN ANALOG, VACUOLAR PROTONE ATP HYDROLASE INHIBITOR, APOTOSIS INDUCER AND ANTICANCER AGENT
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机译:刀豆蛋白类似物,液泡质子ATP水解酶抑制剂,凋亡诱导剂和抗癌剂
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摘要
PROBLEM TO BE SOLVED: To obtain a new compound having V-ATPase-inhibiting activity.;SOLUTION: The new compound is expressed by general formula (I) [wherein R1 expresses H or formula (2)]. A pharmaceutically permissible salt of the same is claimed. A vacuolar protone ATP hydrolase inhibitor, an apotosis inducer and an anticancer agent containing the compound expressed by general formula (I) or its pharmacologically permissible salt are also claimed.;COPYRIGHT: (C)2004,JPO
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