首页> 外国专利> Sildenafil citrate solid dispersions having high water solubility

Sildenafil citrate solid dispersions having high water solubility

机译:具有高水溶性的枸den酸西地那非固体分散体

摘要

Solid dispersions of sildenafil citrate and certain highly water soluble sugars are provided, which solid dispersions significantly increase the water solubility of sildenafil citrate. Methods for preparing highly water soluble solid dispersions of the present invention facilitate the incorporation of sildenafil citrate into new sildenafil citrate containing dosage forms which were heretofore impractical. A method for improving and/or enhancing the sexual response in animals, particularly humans, by administering such new sildenafil citrate containing dosage forms is also provided.
机译:提供了枸den酸西地那非和某些高水溶性糖的固体分散体,该固体分散体显着增加了枸sil酸西地那非的水溶性。制备本发明的高度水溶性固体分散体的方法有助于将枸sil酸西地那非掺入到迄今不切实际的新的含有枸sil酸西地那非的剂型中。还提供了通过施用这种新的含枸sil酸西地那非的剂型来改善和/或增强动物特别是人的性反应的方法。

著录项

  • 公开/公告号AU7354501A

    专利类型

  • 公开/公告日2002-01-30

    原文格式PDF

  • 申请/专利权人 LAVIPHARM LABORATORIES INC.;

    申请/专利号AU20010073545

  • 发明设计人 LI TAO;LI-LAN CHEN;

    申请日2001-07-18

  • 分类号A61K31/495;A61K31/505;

  • 国家 AU

  • 入库时间 2022-08-22 00:39:27

相似文献

  • 专利
  • 外文文献
  • 中文文献
获取专利

客服邮箱:kefu@zhangqiaokeyan.com

京公网安备:11010802029741号 ICP备案号:京ICP备15016152号-6 六维联合信息科技 (北京) 有限公司©版权所有
  • 客服微信

  • 服务号