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New dimeric 1,4-di:hydro-pyridine derivatives are HIV-1 protease inhibitors
New dimeric 1,4-di:hydro-pyridine derivatives are HIV-1 protease inhibitors
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机译:新的二聚1,4-二:氢吡啶衍生物是HIV-1蛋白酶抑制剂
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摘要
Dimeric 1,4-dihydropyridine compounds of formulae (IV), (Va) and (Vb) are new. R1 = H, T, COOT or COT; R2 = COOT' (in (IV) and (Vb)) or HOCH2 (in (Va)); X = OT', OH, CH2OT', H or NH2; T = alkyl or aryl; and T' = alkyl.
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机译:式(IV),(Va)和(Vb)的二聚1,4-二氢吡啶化合物是新的。 R1 = H,T,COOT或COT; R2 = COOT'(在(IV)和(Vb)中)或HOCH2(在(Va)中); X = OT',OH,CH2OT',H或NH2; T =烷基或芳基; T'=烷基。
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