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Compound, composition form of unit dosage methods for administration of a biologically active agent to prepare a composition for administration of an active agent and to prepare a CompoThs and pharmacological composition

机译：用于施用生物活性剂以制备用于施用活性剂的组合物以及制备CompoThs和药理学组合物的单位剂量方法的化合物，组合物形式

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摘要

The present invention provides modified amino acids for delivering active agents, and particularly biologically or chemically active agents. The preferred modified amino acids of the present invention include N-acylated or sulfonated amino acids. These modified amino acids are used as carriers to facilitate the delivery of a cargo to a target. Such modified amino acids are well suited to form non-covalent mixtures with biologically-active agents for oral administration to animals. Methods for the preparation and administration of the modified amino acids and compositions including the same are also provided.

机译：本发明提供了用于递送活性剂，特别是生物或化学活性剂的修饰的氨基酸。本发明优选的修饰氨基酸包括N-酰化或磺化氨基酸。这些修饰的氨基酸用作载体以促进将货物递送至靶标。此类修饰的氨基酸非常适合与生物活性剂形成非共价混合物，以口服施用于动物。还提供了制备和施用修饰的氨基酸的方法以及包括其的组合物。

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公开/公告号BR9604880A

专利类型
公开/公告日1998-05-19

原文格式PDF
申请/专利权人 EMISPHERE TECHNOLOGIES INC.;
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申请/专利号BR19969604880
发明设计人 ANDREA LEONE-BAY;KOC-KAN HO;SAM J. MILSTEIN;JEFFREY BRUCE PRESS;DONALD J. SARUBBI;
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申请日1996-04-01
分类号A61K38/00;C07C53/126;C07C53/134;C07C57/26;C07C57/30;C07C57/42;C07C59/76;C07C59/80;C07C59/84;C07C59/205;C07C229/10;C07C311/19;C07D207/34;C07D213/60;C07D333/30;
国家 BR
入库时间 2022-08-22 02:58:34

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