首页> 外国专利> PHARMACEUTICAL COMPOSITIONS, FOR INHIBITING VASOMOTOR SYMPTOMS AND ATTENDING PSYCHOLOGICAL DISTURBANCES SURROUNDING POST-MENOPAUSAL SYNDROME CONTAINING 2-PHENYL-3-AROYL-BENZOTHIOPHENE DERIVATIVES AND PROCESS FOR THEIR PREPARATION

PHARMACEUTICAL COMPOSITIONS, FOR INHIBITING VASOMOTOR SYMPTOMS AND ATTENDING PSYCHOLOGICAL DISTURBANCES SURROUNDING POST-MENOPAUSAL SYNDROME CONTAINING 2-PHENYL-3-AROYL-BENZOTHIOPHENE DERIVATIVES AND PROCESS FOR THEIR PREPARATION

机译:药物组合物,用于抑制血管痉挛症状,并消除围绕绝经后综合征(包含2-苯基-3-芳基-苯并噻吩衍生物)的心理障碍及其制备方法

摘要

A method of inhibiting vasomotor symptoms and attending psychological disturbances surrounding post-menopausal syndrome comprising administering to a female human in need of treatment an effective amount of a compound having the formula CHEM wherein R1 and R3 are independently hydrogen, -CH3, CHEM wherein Ar is optionally substituted phenyl; R2 is selected from the group consisting of pyrrolidine, hexamethyleneamino, and piperidino; or a pharmaceutically acceptable salt of solvate thereof.
机译:抑制绝经后综合症周围的血管舒缩症状和心理障碍的方法,包括对需要治疗的女性给予有效量的具有式的化合物,其中R 1和R 3独立地为氢,-CH 3,其中Ar是任选取代的苯基; R 2选自吡咯烷,六亚甲基氨基和哌啶子基;或其溶剂化物的可药用盐。

著录项

  • 公开/公告号HUT71478A

    专利类型

  • 公开/公告日1995-11-28

    原文格式PDF

  • 申请/专利权人 ELI LILLY AND CO.;

    申请/专利号HU19940003662

  • 发明设计人 CULLINANGEORGE JOSEPH;

    申请日1994-12-19

  • 分类号A61K31/445;A61K31/40;A61K31/38;

  • 国家 HU

  • 入库时间 2022-08-22 03:53:55

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