首页> 外国专利> PERCUTANEOUS ADMINISTRATION OF SPIRONOLACTONE AS SYSTEMICALLY ACTIVE ANTI-ANDROGEN AND PREPARATION COMPOSITION FOR LOCAL THERAPY OF ACNE VULGARIS, SEBORRHEIC DERMATITIS AND HIRSUTISM

PERCUTANEOUS ADMINISTRATION OF SPIRONOLACTONE AS SYSTEMICALLY ACTIVE ANTI-ANDROGEN AND PREPARATION COMPOSITION FOR LOCAL THERAPY OF ACNE VULGARIS, SEBORRHEIC DERMATITIS AND HIRSUTISM

机译:螺内酯作为全身活性抗雄激素的经皮给药及寻常性痤疮,脂溢性皮炎和湿疹的局部治疗的制剂组成

摘要

PURPOSE: To obtain a spironolactone-contg. preparation composition for application to human skin site(s) suffered from acne, seborrheic symptom or hirsutism for the purpose of the lesion's effective therapy. ;CONSTITUTION: This preparation composition for the local application of spironolactone as active ingredient for the purpose of mitigating androgen activity raised in the skin, comprises a safe and effective amount of spironolactone (at 0.1-10 wt.%), a penetration potentiator containing an N,N-di(lower alkyl)laurinamide and a pharmaceutically acceptable vehicle.;COPYRIGHT: (C)1995,JPO
机译:目的:获得螺内酯。用于治疗痤疮,脂溢性症状或多毛症的人皮肤部位的制剂组合物,用于病变的有效治疗。 ;组成:该制剂组合物用于局部施用螺内酯作为活性成分,目的是减轻皮肤中产生的雄激素活性,包含安全有效量的螺内酯(0.1-10 wt。%),一种渗透增强剂,含有N,N-二(低级烷基)月桂酰胺和药学上可接受的媒介物;版权:(C)1995,JPO

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