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5-2-2-Amino-2-oxoethylmethylaminoethyl-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5(5H)-benzothiazepine-4-one derivatives, their preparation and their use in therapy
5-2-2-Amino-2-oxoethylmethylaminoethyl-2,3-dihydro-3-hydroxy-2-(4-methoxyphenyl)-1,5(5H)-benzothiazepine-4-one derivatives, their preparation and their use in therapy
Compounds, in the form of pure diastereoisomers or of mixtures thereof, corresponding to the general formula (I) IMAGE in which R1 represents a hydrogen atom or a C2-C4 alkanoyl group, R2 represents a hydrogen atom or a C1-C4 alkyl group, n represents a number from 0 to 3 and R3 represents either a phenyl group bearing from 1 to 3 substituents chosen from halogen atoms and trifluoromethyl, methyl, C1-C4 alkoxy or alkylthio, nitro, cyano, carbamoyl, acetamido, methanesulphonamido, methoxycarbonyl or phenylcarbonyl groups, or an aromatic heterocyclic group such as a pyridyl or imidazolyl group. Use in therapy.
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