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首页> 外国专利> NOVEL AMINOISOXAZOLE DERIVATIVE AND REMEDY FOR CEREBROVASCULAR DISORDER COMPRISING SAID DERIVATIVE AS ACTIVE INGREDIENT

NOVEL AMINOISOXAZOLE DERIVATIVE AND REMEDY FOR CEREBROVASCULAR DISORDER COMPRISING SAID DERIVATIVE AS ACTIVE INGREDIENT

机译：新的氨基异恶唑衍生物和补救措施，包括有效衍生物作为有效成分的脑血管疾病。

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PURPOSE:To obtain the titled remedy comprising an aminoisoxazole derivative as a main component. CONSTITUTION:A remedy for cerebrovascular disorder containing a compound shown by the formula (R1 is alkyl, phenyl, benzyl, phenethyl, etc.; R2 is alkyl, cyano, amido, phenyl, etc.; R3 and R4 are H, alkyl, formyl, acetyl, etc., or R3 and R4 are bonded to form morpholino, piperazinyl, piperidyl, etc.) or a salt thereof (e.g. 5-amino-3-phenylisoxazole, etc.) as a main component. The remedy has inhibitory action on brain edema, protecting action on ischemic focus and improving action on nerve symptoms. An injection, suppository or oral drug may be cited as the dosage form. The remedy may be dissolved in 20% glycerol solution and used as a transfusion solution. A preferable dose in an acute phase of cerebrovascular disorder is 0.1-2.0g/day.
机译：目的：获得包含氨基异恶唑衍生物作为主要成分的标题药物。组成：一种用于脑血管疾病的药物，其包含下式所示的化合物（R 1为烷基，苯基，苄基，苯乙基等; R 2为烷基，氰基，酰胺基，苯基等; R 3 R和R 4为H，烷基，甲酰基，乙酰基等，或R 3和R 4结合形成吗啉代，哌嗪基，哌啶基等）或其盐（例如5-氨基-3-苯基异恶唑等）为主要成分。该药物对脑水肿有抑制作用，对缺血性局部具有保护作用，对神经症状有改善作用。剂型可以是注射剂，栓剂或口服药物。可以将药物溶解在20％的甘油溶液中并用作输注溶液。脑血管疾病急性期的优选剂量是0.1-2.0g /天。

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