首页> 外国专利> Di - curly bracket on 2 - aminocyclopent - 1 - s - 1 - thiocarbonyl curly bracket to - disulfides, such as well as a process for the preparation of pharmaceutical compositions containing same

Di - curly bracket on 2 - aminocyclopent - 1 - s - 1 - thiocarbonyl curly bracket to - disulfides, such as well as a process for the preparation of pharmaceutical compositions containing same

机译：2-氨基环戊-1-s-1-硫代羰基大括号内的二-二硫化物的双花括号，以及包含该花括号的药物组合物的制备方法

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摘要

Novel N-substituted 2-amino-cyclopent-1-ene-1-dithiocarboxylic acids of the general formula IMAGE in which R denotes an unsubstituted straight or branched alkyl group having 5 or 6 carbon atoms, an alkyl group having 1 to 6 carbon atoms, which is substituted by alkoxy groups having 1 to 4 carbon atoms, or by hydroxyl, carboxyl and/or amino groups, an alkenyl group having 2 to 4 carbon atoms, a cycloalkyl group having 3 to 8 carbon atoms, or a phenyl group, are prepared by reacting 2-amino-cyclopent-1-ene-1-dithiocarboxylic acid with amines of the general formula NH2-R. The novel compounds have a dopamine- beta -hydroxylase-inhibiting effect.

机译：通式的新型N-取代的2-氨基-环戊-1-烯-1-二硫代羧酸，其中R表示具有5或6个碳原子的未取代的直链或支链烷基，具有1至6的烷基碳原子，该碳原子被具有1-4个碳原子的烷氧基或羟基，羧基和/或氨基，具有2-4个碳原子的烯基，具有3-8个碳原子的环烷基或苯基取代通过使2-氨基-环戊-1-烯-1-二硫代羧酸与通式为NH2-R的胺反应制备基团。新化合物具有多巴胺-β-羟化酶抑制作用。

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公开/公告号DE2758809A1

专利类型
公开/公告日1978-07-06

原文格式PDF
申请/专利权人 RICHTER GEDEON VEGYESZET;
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申请/专利号DE19772758809
发明设计人 MATOLCSY GYOERGY DR HU;BARTOK GEB BERENCSY PIROSKA HU;KISS BELA HU;PALOSI EVA DR HU;KARPATI EGON DR HU;SZPORNY LASZLO DR HU;
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申请日1977-12-30
分类号C07C149/26;A61K31/095;C07C148/00;
国家 DE
入库时间 2022-08-22 21:54:26

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