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new secondary to diazabicyclo (c). undecapentaene and method for preparation of the composition and its salts
new secondary to diazabicyclo (c). undecapentaene and method for preparation of the composition and its salts
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机译：diazabicyclo（c）的新中学。十一碳烯和制备该组合物及其盐的方法
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摘要
1334271 Diazabicycloundecapentane derivative E GY T GYOGYSZERVEGYESZETI GYAR 10 May 1971 [6 Nov 1970] 14045/71 Heading C2C The novel compound I and acid addition salts thereof are prepared (1) by reaction of compounds II with hydrazine or hydrazine hydrate to give compounds III and reacting compounds III with an acid, (2) by reaction of a 1-veratryl-3-methyl-4-ethyl- 6,7 - dimethoxy - isobenzopyrilium salt with hydrazine or hydrazine hydrate, followed by treatment with an acid or (3) by reaction of 3 - (2 - veratroyl - 4,5 - dimethoxyphenyl)- pentan-2-one with hydrazine or hydrazine hydrate in a mixture of one or more 1-4C alcohols and benzene to give an adduct IV which is then decomposed with an acid. Pharmaceutical compositions comprise a compound I together with a suitable excipient and are useful as tranquillizers.
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机译：1334271二氮杂双环庚烷衍生物E GY T GYOGYSZERVEGYESZETI GYAR 1971年5月10日[1970年11月6日] 14045/71标题C2C通过以下方法制备新的化合物I及其酸加成盐（1）：使化合物II与肼或水合肼反应，得到化合物III和使化合物III与酸反应，（2）使1-veratryl-3-甲基-4-乙基-6,7-二甲氧基-异苯并吡喃鎓盐与肼或水合肼反应，然后用酸或（3）处理在一种或多种1-4C醇和苯的混合物中，使3-（2-叔丙基-4,5,5-二甲氧基苯基）-戊烷-2-酮与肼或水合肼反应，生成加合物IV，然后将其分解酸。药物组合物包含化合物I和合适的赋形剂，并且可用作镇静剂。
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