首页> 外国专利> N-Allyl-2-(6-butyl-1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrido2,3-dpyrimidin-5-yl)sulfanylacetamide for treating and preventing anxiety or Neuroinflammatory diseases

N-Allyl-2-(6-butyl-1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrido2,3-dpyrimidin-5-yl)sulfanylacetamide for treating and preventing anxiety or Neuroinflammatory diseases

机译:n-allyl-2 - [(6-丁基-1,3-二甲基-2,4-二氧氧-1,2,3,4-四氢吡啶[2,3-d]嘧啶-5-基)磺酰乙酰乙酰胺治疗和预防焦虑或神经胰腺炎疾病

摘要

The present invention is N-aryl-2-[(6-butyl-1,3-dimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrido[2,3-d]pyrimidine- It relates to a pharmaceutical composition for the prevention and treatment of anxiety disorders or neuroinflammatory diseases containing 5-yl)sulphenyl]acetamide as an active ingredient, and the N-aryl-2-[(6-butyl-1,3) of the present invention -Dimethyl-2,4-dioxo-1,2,3,4-tetrahydropyrido[2,3-d]pyrimidine-5-yl)sulphenyl]acetamide is CHI3L1 (Chitinase 3-like 1) It can be used as a composition for preventing and treating anxiety symptoms or neuro-inflammatory diseases because it binds to inhibit function and relieves nerve inflammation to improve anxiety symptoms.
机译:本发明是N-芳基-2 - [(6-丁基-1,3-二甲基-2,4-二氧氧-1,2,3,4-四氢呋喃[2,3-D]嘧啶 - 它涉及a用于预防和治疗含有5-基)硫烯基的焦虑障碍或神经炎疾病的药物组合物作为活性成分,以及本发明的N-芳基-2- [(6-丁基-1,3) - 二甲基-2,4-二氧基-1,2,3,4-四氢吡啶-5-基)硫烯基]乙酰胺是CHI3L1(几丁质酶3样1),可用作预防的组合物并治疗焦虑症状或神经炎症疾病,因为它结合抑制功能并减轻神经炎症以改善焦虑症状。

著录项

  • 公开/公告号KR102249560B1

    专利类型

  • 公开/公告日2021-05-10

    原文格式PDF

  • 申请/专利权人

    申请/专利号KR1020190117192

  • 发明设计人 홍진태;이희범;

    申请日2019-09-24

  • 分类号A61K31/519;A61P25;A61P25/22;

  • 国家 KR

  • 入库时间 2022-08-24 18:46:57

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