首页> 外国专利> 4 - (1-phenyl-1h - 1,2,3 triazol-4-yl) - sulfamate derivatives of phenol, 4 - (1-phenyl-1h - 1,2,3 triazol-4-yl) - derivatives of phenol, their medical applications And 4 - (1-phenyl-1h - 1,2,3 triazol-4-yl) - Method for obtaining phenylene ruffate derivative

4 - (1-phenyl-1h - 1,2,3 triazol-4-yl) - sulfamate derivatives of phenol, 4 - (1-phenyl-1h - 1,2,3 triazol-4-yl) - derivatives of phenol, their medical applications And 4 - (1-phenyl-1h - 1,2,3 triazol-4-yl) - Method for obtaining phenylene ruffate derivative

机译：4 - （1-苯基-1H - [1,2,3]三唑-4-基） - 苯酚的磺酸盐衍生物，4 - （1-苯基-1H - [1,2,3]三元唑-4-基） - 苯酚，其医疗应用和4 - （1-苯基-1H - [1,2,3]三唑-4-基）的衍生物 - 获得亚苯基鼻芳酸酯衍生物的方法

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The present invention relates to a new compound, 4 - (1-phenyl-1h - [1,2,3] triazol-4-yl) - phenyllafamate derivatives and 4 - (1-phenyl-1h - [1,2,3] triazol-4-yl) - phenol derivatives.The subject matter of the present invention is for medical applications of 4 - (1-phenyl-1h - [1,2,3] triazol-4-yl) - phenyllafate derivatives and 4 - (1-phenyl-1h - [1,2,3] triazole-4-yl) - phenol derivatives.The subject matter of the present invention is the use of a novel compound as a drug having the properties of a steroid sulfatase inhibitor and / or estrogen receptor modulator.The present invention relates to medical applications of novel compounds used as antimicrobial agents and / or estrogen receptor modulators.Specifically, 4 - (1-phenyl-1h - [1,2,3] triazol-4-yl) - phenylsulfamate derivatives are used as medications in the treatment of cancer.The present invention also relates to the preparation process of these new compounds, and 4 - (1-phenyl-1h - [1,2,3] triazol-4-yl) - phenol derivatives are intermediate products obtained by sulfamate derivatives.No selection

机译：本发明涉及新化合物，4 - （1-苯基-1H - [1,2,3]三唑-4-基） - 苯二胺衍生物和4-（1-苯基-1H - [1,2,3 ]三唑-4-基） - 苯酚衍生物。本发明的主题是用于4 - （1-苯基-1H - [1,2,3]三元唑-4-基） - 苯并三唑衍生物和4的医学应用 - （1-苯基-1H - [1,2,3]三唑-4-基） - 苯酚衍生物。本发明的主题是使用一种新化合物作为具有类固醇硫酸酶抑制剂性质的药物的药物和/或雌激素受体调节剂。本发明涉及用作抗微生物剂和/或雌激素受体调节剂的新化合物的医学应用。特异性，4 - （1-苯基-1H - [1,2,3]三唑-4- Y1） - 苯磺酸盐衍生物用作治疗癌症的药物。本发明还涉及这些新化合物的制备方法，4 - （1-苯基-1H - [1,2,3]三唑-4- YL） - 苯酚衍生物是通过磺胺酸酯衍生物获得的中间产物。没有选择

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公开/公告号JP2022501310A

专利类型
公开/公告日2022-01-06

原文格式PDF
申请/专利权人ポリテクニカグダンスカ;
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申请/专利号JP20200570953
发明设计人デムコビック;セバスチャン;ダスコ;マテウシュ;レイション;ヤーヌシュ;
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申请日2018-08-20
分类号C07D249/06;A61K31/4192;A61P35;A61P31/04;A61P5/32;A61P43;
国家 JP
入库时间 2022-08-24 23:15:58

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