Synthesis, characterization and biological activity of benzothiazoles derivatives

机译：苯并噻唑衍生物的合成，表征和生物活性

获取原文

页面导航

摘要
著录项
相似文献
相关主题

摘要

In the present investigation 2-(hydrazinylmethyl)-1,3-benzothiazole was reacted with aryl aldehyde to give 2-{[2Z)-2-arylhydrazinyl]methyl}-1,3-benzothiazole (3a-f), which in absolute ethanol treated with thioglycolic acid (0.001 mol) and anhydrous zinc chloride under reflux for 8 hr to get 3-[1,3-benzothiazol-2-ylmethyl) amino]-5-(aryl)-1,3-thiazolidin-2-ones (4a-f). On the other hand [Benzothiozole N-aryl thiozolemethanamines] (5a-f) were obtained, when the compounds (3a-f), are treated with diazomethane.

机译：在本发明的研究中，将2-（肼基甲基）-1,3-苯并噻唑与芳基醛反应，得到2 - {[2z）-2-芳基肼基]甲基} -1,3-苯并噻唑（3A-F），这是绝对的在回流下用巯基乙酸（0.001mol）和无水氯化锌处理的乙醇，得到8小时，得到3- [1,3-苯并噻唑-2-基甲基）氨基] -5-（芳基）-1,3-噻唑烷-2- 那些（4A-F）。另一方面，当化合物（3A-F）处理用重氮甲烷处理时，得到苯并噻唑N-芳基甲基甲酰胺]（5A-F）。

著录项

来源
《International Conference on Physics of Materials and Nanotechnology》|2020年|various paging|共4页
会议地点
作者
Pathki Uma; Firasath Unnisa; Pallati Naresh; Sai Prakash; P. R. Sushma; Kamatala Chinna Rajanna;
展开▼
作者单位

展开▼
会议组织
原文格式 PDF
正文语种
中图分类 TB3-53;
关键词

相似文献

外文文献
中文文献
专利

1. Synthesis, Characterization and Biological Activities of Mercury(II) Ternary Complexes of 2-Substituted Benzothiazoles Derivatives [J] . Manmohan Singh Chauhan, Mitlesh Kumari Yadav, Aruna Sharma Asian Journal of Chemistry: An International Quarterly Research Journal of Chemistry . 2018,第8期

机译：2-取代苯并噻唑衍生物的汞（II）三元复合物的合成，表征和生物活性
2. Design, synthesis, spectral characterization, DNA interaction and biological activity studies of copper(II), cobalt(II) and nickel(II) complexes of 6-amino benzothiazole derivatives [J] . Daravath Sreenu, Kumar Marri Pradeep, Rambabu Aveli, Journal of Molecular Structure . 2017,第期

机译：6-氨基苯并噻唑衍生物的铜（II），钴（II），钴（II）和镍（II）络合物的设计，合成，光谱表征，DNA相互作用及生物活性研究
3. Novel synthesis and biological activity of 2-substituted derivatives of 3-cyano-4-imino-2-methylthio-8-methoxy-4H-pyrimido[2,1-b][1,3]benzothiazole and 3-amino-4-imino-8-methoxy-2H - Pyrazolo[3′,4′:4,5]pyrimido[2,1-b][1, 3]benzothiazole [J] . Badne S.G., Swamy D.K., Bhosale V.N., Journal of Heterocyclic Chemistry: The International Journal of Heterocyclic Chemistry . 2011,第4期

机译：3-氰基-4-亚氨基-2-亚甲基-2-甲硫基-8-甲氧基-4H-嘧啶基[2,1-b] [1,3]苯并噻唑和3-氨基-4-基团的2-取代衍生物的合成和生物活性亚氨基-8-甲氧基-2H-吡唑并[3'，4'：4,5]嘧啶[2,1-b] [1，3]苯并噻唑
4. Synthesis, characterization and biological activity of benzothiazoles derivatives [C] . Pathki Uma, Firasath Unnisa, Pallati Naresh, International Conference on Physics of Materials and Nanotechnology . 2020

机译：苯并噻唑衍生物的合成，表征和生物活性
5. Design, synthesis, and structure-activity relationship investigation of 3',4'-disubstituted pyranochromone derivatives with diverse biological activities [D] . Zhou, Ting 2010

机译：具有多种生物活性的3'，4'-二取代吡喃并发色酮衍生物的设计，合成及构效关系研究
6. Design synthesis and biological evaluation of novel 1H-124-triazole benzothiazole and indazole-based derivatives as potent FGFR1 inhibitors viafragment-based virtual screening [O] . Jian Liu, Yu Wen, Lina Gao, 2020

机译：通过基于片段的虚拟筛选设计新型1H-124-三唑苯并噻唑和吲唑基衍生物作为强效FGFR1抑制剂的设计合成和生物学评估
7. Synthesis, Characterization and Biological Evaluation of Some Benzothiazole Derivatives as Potential Antimicrobial Agent. [O] . Ashok G. Awale 2016

机译：一些苯并噻唑衍生物作为潜在抗微生物剂的合成，表征及生物学评价。

Synthesis, characterization and biological activity of benzothiazoles derivatives

摘要

著录项

相似文献

相关主题

期刊订阅