Synthesis and Biological Activity of New Pyrethroid Acid Oxime-esters Containing Pyrazole Ring

MA Jun-an; HUANG Run-qiu; FENG Lei; SONG Jian QIU De-wen

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Synthesis and Biological Activity of New Pyrethroid Acid Oxime-esters Containing Pyrazole Ring

机译：新型含吡唑环的拟除虫菊酯肟酯的合成及生物活性

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A series of compounds containing oxime-ester linkage and pyrazole ring (in place of the ester linkage and the alcohol moiety in pyrethroid ester) was designed and synthesized. The structures of all the compounds prepared were confirmed by ~1H NMR and MS spectroscopy as well as elemental analyses. The bioassay data of those compounds against tobacco mosaic virus (TMV), cucumber mosaic virus (CMV). potato virus X (PVX) and potato virus Y(PVY) were presented. Among them compound 6i was found to possess significant plant antiviral activities. But all the compounds showed low insecticidal and acaricidal activities.

机译：设计并合成了一系列含有肟酯键和吡唑环的化合物（取代了拟除虫菊酯中的酯键和醇部分）。制备的所有化合物的结构均通过〜1 H NMR和MS光谱以及元素分析得到证实。这些化合物针对烟草花叶病毒（TMV），黄瓜花叶病毒（CMV）的生物测定数据。介绍了马铃薯病毒X（PVX）和马铃薯病毒Y（PVY）。其中化合物6i被发现具有重要的植物抗病毒活性。但是所有化合物均显示出较低的杀虫和杀螨活性。

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来源
《Chemical Research in Chinese Universities》 |2003年第3期|p.297-301|共5页
作者
MA Jun-an; HUANG Run-qiu; FENG Lei; SONG Jian QIU De-wen;
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作者单位

Institute and State Key Laboratory of Elemento-organic Chemistry, Nankai University, Tianjin 300071, P. R. China;

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原文格式 PDF
正文语种 eng
中图分类化学;
关键词
pyrethroid; oxime-ester; synthesis; pyrazole; plant antiviral activity;

机译：拟除虫菊酯;肟酯;合成;吡唑;植物抗病毒活性;

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1. Synthesis and Biological Activity of New Pyrethroid Acid Oxime-esters Containing Pyrazole Ring [J] . MA Jun-an, HUANG Run-qiu, FENG Lei, 高等学校化学研究（英文版） . 2003,第003期

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Synthesis and Biological Activity of New Pyrethroid Acid Oxime-esters Containing Pyrazole Ring

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