Synthesis of β-alkoxy-N-protected phenethylamines via one-pot copper-catalyzed aziridination and ring opening

Jorge Saavedra-Olavarría; Matías Madrid-Rojas; Iriux Almodovar; Patricio Hermosilla-Ibá?ez; Edwin G. Pérez

首页> 外文期刊>RSC Advances >Synthesis of β-alkoxy-N-protected phenethylamines via one-pot copper-catalyzed aziridination and ring opening

【24h】

Synthesis of β-alkoxy-N-protected phenethylamines via one-pot copper-catalyzed aziridination and ring opening

机译：一锅铜催化的叠氮化和开环反应合成β-烷氧基-N-保护的苯乙胺

获取原文

掌桥外文数据库（机构版） >>

开具论文收录证明 >>

文献代查 >>

页面导航

摘要
著录项
相似文献
相关主题

摘要

A regioselective, copper-catalyzed, one-pot aminoalkoxylation of styrenes using primary and secondary alcohols and three different iminoiodanes as alkoxy and nitrogen sources respectively, is reported. The β-alkoxy- N -protected phenethylamines obtained were used to synthesise β-alkoxy- N -benzylphenethylamines which are interesting new compounds that could act as possible neuronal ligands.

机译：报道了分别使用伯醇和仲醇以及三种不同的亚氨基碘酮作为烷氧基和氮源的苯乙烯的区域选择性，铜催化的一锅氨基氨基烷氧基化反应。将获得的β-烷氧基-N-保护的苯乙胺用于合成β-烷氧基-N-苄基苯乙胺，这是有趣的新化合物，可以充当可能的神经元配体。

著录项

来源
《RSC Advances》 |2018年第49期|共5页
作者
Jorge Saavedra-Olavarría; Matías Madrid-Rojas; Iriux Almodovar; Patricio Hermosilla-Ibá?ez; Edwin G. Pérez;
展开▼
作者单位

展开▼
收录信息
原文格式 PDF
正文语种
中图分类化学;
关键词

相似文献

外文文献
中文文献
专利

1. Synthesis of β-alkoxy-N-protected phenethylamines via one-pot copper-catalyzed aziridination and ring opening [J] . Jorge Saavedra-Olavarría, Matías Madrid-Rojas, Iriux Almodovar, RSC Advances . 2018,第49期

机译：一锅铜催化的叠氮化和开环反应合成β-烷氧基-N-保护的苯乙胺
2. Synthesis of beta-alkoxy-N-protected phenethylamines via one-pot copper-catalyzed aziridination and ring opening [J] . Saavedra-Olavarria Jorge, Madrid-Rojas Matias, Almodovar Iriux, RSC Advances . 2018,第49期

机译：通过单盆铜催化的叠氮化和环开口合成β-烷氧基-N保护的苯乙胺
3. Metal-free synthesis of 1,2-amino alcohols by one-pot olefin aziridination and acid ring-opening [J] . Hua Yong-Gang, Yang Qian-Qian, Yang Yi, Tetrahedron letters: The International Journal for the Rapid Publication of Preliminary Communications in Organic Chemistry . 2018,第28期

机译：1,2-氨基醇的无金属合成1-壶烯烃叠氮化和酸环开环
4. One-pot Synthesis of 10-Membered Ring Cyclophanes:Size-Controlled Macrocyclization via Cyano-Gilman Cuprate [C] . MoWu.Yoshihiro, Miyakeand Masahiko Symposium on Organometallic Chemistry . 2003

机译：10元环环烷的单壶合成：通过Cyano-Gilman铜替代铜尺寸控制的宏次数
5. Part I. One-pot synthesis of secondary alcohols and one-pot asymmetric synthesis of secondary propargylic alcohols. Part II. Redox isomerization of secondary propargylic alcohols to enones. Part III. Synthesis study towards C9-C14 fragment of (+)-discodermolide. Part IV. Asymmetric synthesis of anti, anti-stereotriad building blocks for polypropionate natural products [D] . Xie, Qiuzhe 2007

机译：第一部分：仲醇的一锅法合成和仲炔丙醇的一锅法不对称合成。第二部分仲炔丙醇的氧化还原异构化为烯酮。第三部分（+）-discodermolide C9-C14片段的合成研究。第四部分聚丙烯酸酯天然产物的抗，抗立体三环构建基的不对称合成
6. One-pot stereoselective synthesis of αβ-differentiated diamino esters via the sequence of aminochlorination aziridination and intermolecular SN2 reaction [O] . Yiwen Xiong, Ping Qian, Chenhui Cao, 2014

机译：通过氨基氯化叠氮化和分子间SN2反应的序列一锅立体选择性合成αβ-差异化的二氨基酯
7. Synthesis of β-alkoxy-N-protected phenethylamines via one-pot copper-catalyzed aziridination and ring opening [O] . Jorge Saavedra-Olavarría, Matías Madrid-Rojas, Iriux Almodovar, 2018

机译：通过单盆铜催化的叠氮化和环开口合成β-烷氧基-N保护的苯乙胺

Synthesis of β-alkoxy-N-protected phenethylamines via one-pot copper-catalyzed aziridination and ring opening

摘要

著录项

相似文献

相关主题

期刊订阅