Synthesis of 3-substituted pyrrolidines

A. V. Kurkin; E. A. Sumtsova; M. A. Yurovskaya

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Synthesis of 3-substituted pyrrolidines

机译：3-取代的吡咯烷的合成

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摘要

A method was developed for the synthesis of derivatives of 3-substituted pyrrolidines from activated alkenes by 1,3-dipolar cycloaddition of unstable 2-benzylazomethylide, generated in situ from N-benzyl-N-(methoxymethyl)-N-(trimethylsilyl)amine. A method was developed for the reduction of 4-(3-pyrrolidyl)pyridine, prepared by the above-mentioned method, to the corresponding derivatives of (3-pyrrolidyl)piperidine with high yields under mild conditions.

机译：开发了一种方法，用于由活化的烯烃通过不稳定的2-苄基偶氮亚甲基的1，3-偶极环加成反应从活化的烯烃合成3-取代的吡咯烷衍生物，所述不稳定的2-苄基偶氮甲基化物是由N-苄基-N-（甲氧基甲基）-N-（三甲基甲硅烷基）胺生成的。开发了一种在温和条件下以高收率将通过上述方法制备的4-（3-吡咯烷基）吡啶还原为相应的（3-吡咯烷基）哌啶衍生物的方法。

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《Chemistry of heterocyclic compounds》 |2007年第1期|共7页
作者
A. V. Kurkin; E. A. Sumtsova; M. A. Yurovskaya;
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正文语种 eng
中图分类杂环化合物;
关键词
N-benzyl-N-(methoxymethyl)-N-(trimethylsilylmethyl)amine; piperidines; reduction of pyridines; 1; 3-dipolar cycloaddition to alkenes;

机译：N-苄基-N-（甲氧基甲基）-N-（三甲基硅烷基甲基）胺;哌啶;吡啶的还原;1;3-偶极环加成烯烃;

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1. An enantioselective approach to 3-substituted pyrrolidines: Asymmetric synthesis for pyrrolidine core of serotonin norepinephrine reuptake inhibitors (SNRIs) [J] . Garg Yuvraj, Sharma Pooja, Pandey Satyendra Kumar Tetrahedron letters: The International Journal for the Rapid Publication of Preliminary Communications in Organic Chemistry . 2017,第36期

机译：3取代吡咯烷的对映选择性方法：羟色素核肾上腺素再摄取抑制剂（SNRIS）的吡咯烷核心的不对称合成
2. SYNTHESIS OF NOVEL ANTIMICROBIAL DERIVATIVES OF 3-SUBSTITUTED PYRROLIDINE2, 5-DIONES USING PHARMACOPHORE HYBRID APPROACH: PART-I [J] . SMITA PAWAR, SANJAY SAWANT, AMIT NERKAR, International Journal of Pharmacy and Pharmaceutical Sciences . 2014,第2期

机译：药物-杂合法合成3-取代的吡咯烷2,5-二酮类新型抗菌衍生物
3. Using heteroaryl-lithium reagents as hydroxycarbonyl anion equivalents in conjugate addition reactions with (S, S)-(+)-pseudoephedrine as chiral auxiliary; Enantioselective synthesis of 3-substituted pyrrolidines [J] . Alonso B., Ocejo M., Carrillo L., The Journal of Organic Chemistry . 2013,第2期

机译：在（S，S）-（+）-伪麻黄碱作为手性助剂的共轭加成反应中，使用杂芳基-锂试剂作为羟羰基阴离子当量; 3-取代的吡咯烷的对映选择性合成
4. Synthesis, Characterization and bulk crystal growth of nonlinear 3-substituted salicylidene aniline derivatives [C] . K. Bhat, T. Gebre, A. K. Batra, Conference on Linear and Nonlinear Optics of Organic Materials III; Aug 4-6, 2003; San Diego, California, USA . 2003

机译：非线性3-取代水杨基苯胺衍生物的合成，表征和体相生长
5. Novel palladium-catalyzed synthesis of 3-substituted indoles and its application toward the total synthesis of indolactam V. [D] . Turner, Michael Robert. 2000

机译：3-取代的吲哚的新型钯催化合成及其在吲哚内酰胺V的全合成中的应用
6. Synthesis of 3-Substituted Pyrrolidines via Palladium-Catalyzed Hydroarylation [O] . Joseph B. Sweeney, Julien Doulcet, Bimod Thapa 2018

机译：钯催化的氢芳基化反应合成3-取代的吡咯烷
7. Synthesis of 3-Substituted Pyrrolidines via Palladium-Catalyzed Hydroarylation [O] . Joseph B. Sweeney, Julien Doulcet, Bimod Thapa 2018

机译：通过钯催化的水红合成3取代的吡咯烷

Synthesis of 3-substituted pyrrolidines

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