A facile one pot synthesis of novel N1-(2-nitrophenyl sulphenyl substituted) pyrrolidino[2,1-c][1,4]-benzodiazepine,thiazolidino[3,2-c][1,4]-benzodiazepine andthiazolidino[4,3-c][1,4]-benzodiazepine from the corresponding N-substitutedisatoic anhydride

Sumitra Nain; Varini Gupta; Megha Arya

首页> 外文期刊>Journal of the Indian Chemical Society >A facile one pot synthesis of novel N1-(2-nitrophenyl sulphenyl substituted) pyrrolidino[2,1-c][1,4]-benzodiazepine,thiazolidino[3,2-c][1,4]-benzodiazepine andthiazolidino[4,3-c][1,4]-benzodiazepine from the corresponding N-substitutedisatoic anhydride

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A facile one pot synthesis of novel N1-(2-nitrophenyl sulphenyl substituted) pyrrolidino[2,1-c][1,4]-benzodiazepine,thiazolidino[3,2-c][1,4]-benzodiazepine andthiazolidino[4,3-c][1,4]-benzodiazepine from the corresponding N-substitutedisatoic anhydride

机译：新型N1-（2-硝基苯基亚磺酰基取代的）吡咯烷并[2,1-c] [1,4]-苯并二氮杂，噻唑烷并[3,2-c] [1,4]-苯并二氮杂和噻唑并[4]相应的N-取代的ISA酸酐形成的-，3-c] [1,4]-苯并二氮杂

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A facile one pot synthesis of N1-(2-nitrophenyl sulphenyl substituted) pyrrolidino[2,1-c][1,4]-benzodiazepine (6), 4'-hydroxypyrrolidino[2,l-c][1,4]-benzodiazepine (7), thiazolidino[3,2-c][1,4]-benzodiazepine (8) and thiazolidino[4,3-c][1,4]-benzodiazepine (9) from the reaction of N,-(2-nitrophenyl sulphenyl) isatoic anhydride (1) with L-proline (2), 4-hydroxy-L-proline (3), thiazolidine-2-carboxylic acid (4) and thiazolidinc-3-carboxylic acid (5) respectively has been described. The formation of 6, 7, 8 and 9 from 2, 3, 4 and 5 respectively is believed to take place through the intermediate N-(2-nitrophenyl sulphenyl)-iminoketene (10).

机译：N1-（2-硝基苯基亚磺酰基取代的）吡咯烷并[2,1-c] [1,4]-苯并二氮杂（6），4'-羟基吡咯烷并[2，lc] [1,4]-苯并二氮杂的一锅合成（7）由N，-（2）反应生成的噻唑烷[3,2-c] [1,4]-苯并二氮杂（8）和噻唑烷[4,3-c] [1,4]-苯并二氮杂（9） -硝基苯基亚磺酰基）（1）与L-脯氨酸（2），4-羟基-L-脯氨酸（3），噻唑烷-2-羧酸（4）和噻唑烷-3-羧酸（5）描述。据信分别由2、3、4和5形成6、7、8和9是通过中间体N-（2-硝基苯基亚磺酰基）-亚氨基乙烯酮（10）进行的。

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《Journal of the Indian Chemical Society》 |2009年第9期|共5页
作者
Sumitra Nain; Varini Gupta; Megha Arya;
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正文语种 eng
中图分类化学;
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N1-Substituted-1; 4-benzodiazepines; pyrrolidino- and thiazolidino-1; 4-benzodiazepines; N-(2-nitrophenyl sulphenyl)isatoic anhydride;

机译：N1-取代的[[1;4]-苯并二氮杂;吡咯烷和噻唑烷-[1;4]-苯并二氮杂;N-（2-硝基苯硫基）乙酸酐;

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1. A facile one pot synthesis of novel N1-(2-nitrophenyl sulphenyl substituted) pyrrolidino[2,1-c][1,4]-benzodiazepine,thiazolidino[3,2-c][1,4]-benzodiazepine andthiazolidino[4,3-c][1,4]-benzodiazepine from the corresponding N-substitutedisatoic anhydride [J] . Sumitra Nain, Varini Gupta, Megha Arya Journal of the Indian Chemical Society . 2009,第9期

机译：新型N1-（2-硝基苯基亚磺酰基取代的）吡咯烷并[2,1-c] [1,4]-苯并二氮杂，噻唑烷并[3,2-c] [1,4]-苯并二氮杂和噻唑并[4]相应的N-取代的ISA酸酐形成的-，3-c] [1,4]-苯并二氮杂
2. Synthesis of new aromatic pyrrolo(2,1-c) (1,4)benzodiazepines and pyrrolo(1,2-a)thieno(3,2-e) (1,4)diazepines as anti-tumoral agents. [J] . Lisowski V, Fabis F, Pierre A, Journal of enzyme inhibition and medicinal chemistry. . 2002,第6期

机译：合成新的芳香吡咯并（2,1-c）（1,4）苯并二氮杂和吡咯并（1,2-a）噻吩并（3,2-e）（1,4）二氮杂作为抗肿瘤剂。
3. Efficient synthesis of 3-hydroxy-1,4-benzodiazepines oxazepam and lorazepam by new acetoxylation reaction of 3-position of 1,4-benzodiazepine ring [J] . Cepanec I, Litvic M, Pogorelic I Organic process research & development . 2006,第6期

机译：通过1,4-苯并二氮杂ring环3位的新乙酰氧基化反应有效合成3-羟基-1,4-苯并二氮杂和劳拉西m
4. Solid phase synthesis of 4-methylcarboxy-1,4-benzodiazepine-2,5-diones as building blocks for peptide synthesis [C] . Pascal Verdie, Jean Martinez, Gilles Subra International Peptide Symposium;European Peptide Symposium . 2005

机译：4-甲基羧基-1,4-苯并二氮杂卓-2,5-致肽合成的结构块的固相合成
5. I. PREPARATION AND PROPERTIES OF ALKYL AND ARYL SUBSTITUTED THIOQUINAZOLINES AND SULFOXIDES. II. AN INVESTIGATION OF THE QUINAZOLINE 3-OXIDE-1,4-BENZODIAZEPINE 4-OXIDE REARRANGEMENT. [D] . KUCHAR, MARVIN C. J. 1964

机译：I.烷基和芳基取代的噻喹唑啉和磺胺氧化物的制备和性质。二。喹唑啉3-氧化物-1,4-苯并二氮杂4-氧化物重排的研究。
6. 4-Acetyl-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine [O] . Qing-Jie Zhao, Zheng Liu, Jin Zheng, 2015

机译：4-乙酰基-2,3,4,5-四氢-1H-1,4-苯并二氮杂
7. Pyrimidine-Fused 1,4-Benzodiazepines. Reaction of 1,4-Benzodiazepines with Formamide–POCl3 [O] . Shigeru Kobayashi 1975

机译：嘧啶融合的1,4-苯二氮卓类药物。用甲酰胺-POCl3反应1,4-苯并二氮杂胺

A facile one pot synthesis of novel N1-(2-nitrophenyl sulphenyl substituted) pyrrolidino[2,1-c][1,4]-benzodiazepine,thiazolidino[3,2-c][1,4]-benzodiazepine andthiazolidino[4,3-c][1,4]-benzodiazepine from the corresponding N-substitutedisatoic anhydride

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