Synthesis and Fungicidal Activity of Novel 2,5-Disubstituted-1,3/4-oxadiazole Derivatives

Zi-Ning Cui; Yan-Xia Shi; Li Zhang

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Synthesis and Fungicidal Activity of Novel 2,5-Disubstituted-1,3/4-oxadiazole Derivatives

机译：新型2,5-二取代-1,3 / 4-恶二唑衍生物的合成及杀真菌活性

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A novel series of 1,3,4-oxadiazole derivatives containing a 5-phenyl-2-furan moiety were synthesized from the intermediates diacylhydrazine 3 and acylhydrazone 5 via an efficient approach under microwave irradiation in good yields. Their structures were characterized by IR, ~1H NMR, and elemental analysis. The antifungal tests indicated that the title compounds showed in vivo fungicidal activity against Botrytis cinerea and Rhizoctonia solanii at 500 μg/mL obviously. Some tested compounds even had a superiority effect over the commercial fungicides 40% Pyrimethanil SC and 3% Validamycin AS. The activity between the title compound and their precursors diacylhydrazine 3 and acylhydrazone 5 was also compared and discussed.

机译：通过中间体二酰基肼3和酰基hydr 5的有效方法，在微波辐射下以高收率合成了一系列含有5-苯基-2-呋喃部分的1,3,4-恶二唑衍生物。通过IR，〜1H NMR和元素分析对它们的结构进行了表征。抗真菌试验表明，该标题化合物在500μg/ mL下对灰葡萄孢和番茄红枯病具有明显的体内杀真菌活性。某些测试化合物甚至比40％的嘧霉胺SC和3％的有效霉素AS的商业杀菌剂具有优越的作用。还比较并讨论了标题化合物与其前体二酰基肼3和酰基hydr 5之间的活性。

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《Journal of Agricultural and Food Chemistry》 |2012年第47期|共8页
作者
Zi-Ning Cui; Yan-Xia Shi; Li Zhang;
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2; 5-disubstituted-1; 3; 4-oxadiazole; S-phenyl-2-furan; fungicidal activity; microwave irradiation; synthesis;

机译：2;5-二取代-1;3;4-恶二唑;S-苯基-2-呋喃;杀菌活性;微波辐射;合成;

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1. Synthesis and Fungicidal Activity of Novel 2,5-Disubstituted-1,3/4-oxadiazole Derivatives [J] . Zi-Ning Cui, Yan-Xia Shi, Li Zhang Journal of Agricultural and Food Chemistry . 2012,第47期

机译：新型2,5-二取代-1,3 / 4-恶二唑衍生物的合成及杀真菌活性
2. Synthesis of Some Novel 2,5-Disubstituted 1,3,4-Oxadiazole Derivatives as Potential Antibacterial and Anti-inflammatory activity [J] . Nupur Jaiswal, Arvind Kr. Singh Asian journal of research in chemistry . 2013,第2期

机译：一些新型的2,5-二取代的1,3,4-恶二唑衍生物的合成具有潜在的抗菌和抗炎活性
3. Synthesis and Evaluation of In Vivo Anticonvulsant Activity of 2,5- Disubstituted-1,3,4-Oxadiazole Derivatives [J] . Kikkeri P. Harish, Kikkeri N. Mohana, Lingappa Mallesha, Letters in drug design & discovery . 2013,第8期

机译：2,5-二取代-1,3,4-恶二唑衍生物的体内抗惊厥活性的合成与评价
4. Synthesis and Biological Activity of a 3,5-Disubstituted-1,2,4-Oxadiazole Fungicide Containing 3-Pyrazole Group [C] . Mingming Zhang, Huanqi Cui, Junjun Han, 2019 4th International Conference on Life Sciences, Medicine, and Health（ 2019年第四届生命科学、医学和健康国际会议）（ICLSMH 2019）论文集 . -1

机译：3,5-二取代的-1,2,4-二唑胺含3-吡唑基团的合成和生物活性
5. THE SYNTHESIS AND CHEMICAL REACTIVITY OF THE S-OXIDES OF THIOUREA AND ITS MONO- AND 1,3-DISUBSTITUTED DERIVATIVES (UREA) [D] . BISCHOFF, JUDITH J. 1987

机译：硫脲及其单-和1,3-二取代衍生物（脲）的S-氧化物的合成和化学反应性
6. Synthesis and fungicidal activity of novel 25-disubstituted-134- thiadiazole derivatives containing 5-phenyl-2-furan [O] . Zi-Ning Cui, Ya-Sheng Li, De-Kun Hu, -1

机译：含5-苯基-2-呋喃的新型25-二取代-134-噻二唑衍生物的合成及杀真菌活性
7. Synthesis and fungicidal activity of novel 2,5-disubstituted-1,3,4- thiadiazole derivatives containing 5-phenyl-2-furan [O] . Zi-Ning Cui, Ya-Sheng Li, De-Kun Hu, 2016

机译：新型2,5二取代-1,3,4-噻二唑衍生物的合成和杀菌活性含有5苯基-2-呋喃
8. Liquid Crystalline Polymers Containing Heterocycloalkane Mesogenic Groups. 5. Synthesis of Biphasic Chiral-Smectic Polysiloxanes Containing 2,5-Disubstituted-1,3-Dioxane and 2,5-Disubstituted-1,3,2-Dioxaborinane Based Mesogenic Gr [R] . Hahn, B., Percec, V. 1987

机译：含有杂环烷烃介晶基团的液晶聚合物。 5.含有2,5-二取代-1,3-二恶烷和2,5-二取代-1,3,2-二氧杂硼烷基中间介晶Gr的双相手性 - 近晶聚硅氧烷的合成

Synthesis and Fungicidal Activity of Novel 2,5-Disubstituted-1,3/4-oxadiazole Derivatives

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