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机译:
机译:6-[(3 s,4 s)-4-methyl-1-(pyrimidin-2-ylmethyl)pyrrolidin-3-yl] -1-(tetrahydro-2 h -pyran-4-yl)-的设计和发现1,5-二氢-4 h-吡唑并[3,4- d]嘧啶-4-酮(PF-04447943),一种选择性的脑渗透性pde9a抑制剂,用于治疗认知障碍
机译:Discovery of {1-(4-(2-{hexahydropyrrolo(3,4-c)pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin- 1-yl)cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: design, synthesis, and structure-activity relationships.
机译:发现((1,2,4-oxadiazol-5-yl)pyrrolidin-3-yl)ureidyl衍生物作为G蛋白偶联胆汁酸受体1的选择性非甾体激动剂
机译:双金属成孔剂:3,3-(2-羟基丙烷-1,3-二基)双(Azan-1yl-1-亚烷基)双(2-(4-烷氧基苯基)prop-1-en-1的铜配合物的合成和介晶性质-ol)
机译:DDAH样酶的体内活性探针4-[(2-氯乙亚胺嘧啶基)甲基-N-(prop-2-yn-1-yl)苯甲酰胺的合成
机译:发现((124-oxadiazol-5-yl)pyrrolidin-3-yl)ureidyl衍生物作为G蛋白偶联胆汁酸受体1的选择性非甾体激动剂
机译:catena-poly [[[bis(methanol - Δ)bis(selenocyanate - N)manganese(II)] - γ-1,2-bis(pyridin-4-yl)乙烷 - κ 2N:N′] 1,2-双(吡啶-4-基)乙烷单溶剂化物]
机译:在具有2-卤-1-(Trisubstitu tedcarbomonocycle)-4-烷基-α-(Disubstit utedcarbomonomoncle)-Heteromonocycle-methanol的大鼠中的发育毒性研究的结果。