首页> 外国专利> SUBSTITUTED (4'-HYDROXYPHENYL)CYCLOALKANE AND (4'-HYDROXYPHENYL)CYCLOALKENE COMPOUNDS AND USES THEREOF AS SELECTIVE AGONISTS OF THE ESTROGEN RECEPTOR BETA ISOFORM FOR ENHANCED MEMORY CONSOLIDATION

SUBSTITUTED (4'-HYDROXYPHENYL)CYCLOALKANE AND (4'-HYDROXYPHENYL)CYCLOALKENE COMPOUNDS AND USES THEREOF AS SELECTIVE AGONISTS OF THE ESTROGEN RECEPTOR BETA ISOFORM FOR ENHANCED MEMORY CONSOLIDATION

机译:取代的(4'-羟基苯)环烷烃和(4'-羟基苯)环烯烃化合物,并用作选择性受体激动剂的β-受体异构体,用于增强内存固结

摘要

Disclosed are substituted (4'-hydroxylphenyl)cycloalkane compounds and substituted (4'-hydroxylphenyl)cycloalkene compounds and there use as selective agonists of the estrogen receptor beta isoform (ERβ). The disclosed compounds may be formulated as pharmaceutical compositions and administered for treating diseases associated with ER activity, such as neurological, psychiatric, and/or cell proliferative diseases and disorders as well as for enhancing memory consolidation in subjects in need thereof.
机译:公开了取代的(4'-羟基苯基)环链烷化合物和取代的(4'-羟基苯基)环链烷化合物,并用作雌激素受体β同工型(ERβ)的选择性激动剂。所公开的化合物可以配制成药物组合物,并用于治疗与ER活性有关的疾病,例如神经,精神病和/或细胞增生性疾病和病症,以及用于增强有此需要的受试者的记忆巩固。

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