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TERPENOID ANALOGS FOR TREATING ELECTRICAL DISORDERS IN CENTRAL NERVOUS SYSTEM AND PERIPHERAL NERVOUS SYSTEM AND USES THEREOF

机译：用于治疗中枢神经系统和周围神经系统的电异常的三叉神经类似物及其用途

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摘要

PROBLEM TO BE SOLVED: To provide terpenoid analogs for treating pain, and to provide a method of using the same with the aim of treating pain.SOLUTION: A method for treating electrical disorders in the central nervous system and peripheral nervous system comprises administering into animals (excluding humans) a therapeutically effective amount of a terpene analogue represented by the following formula or a pharmaceutically acceptable salt thereof[Y is an unsubstituted C1-C20 alkylene group, C=O or the like; X is N-(R2) 2 or a substituted C1-C20 alkyl group; R1 is H, a substituted/unsubstituted C1-C20 alkyl group or a substituted/unsubstituted CH-aryl; R2 is each independently H, a substituted/unsubstituted C1-C20 alkyl group, an aryl group, OR, CN, or C(=O) R; R 3 is a substituted/unsubstituted C1-C20 alkyl group substituted/unsubstituted aryl group; W is an unsubstituted C1-C20 alkyl group or an unsubstituted aryl group.]SELECTED DRAWING: None

机译：解决的问题：提供用于治疗疼痛的萜类化合物类似物，并提供用于治疗疼痛的方法。解决方案：用于治疗中枢神经系统和周围神经系统的电障碍的方法包括向动物给药（人类除外）由下式表示的治疗有效量的萜烯类似物或其药学上可接受的盐[Y是未取代的C 1 -C 20亚烷基，C ＝ O等; X为N-（R 2）2或取代的C1-C20烷基。 R1是H，取代/未取代的C1-C20烷基或取代/未取代的CH-芳基; R2分别独立地为H，取代/未取代的C1-C20烷基，芳基，OR，CN或C（= O）R; R 3为取代/未取代的C1-C20烷基取代/未取代的芳基; W是未取代的C1-C20烷基或未取代的芳基。]

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公开/公告号JP2017008076A

专利类型
公开/公告日2017-01-12

原文格式PDF
申请/专利权人 NEUROQUEST INC;
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申请/专利号JP20160154978
发明设计人 MARK A REED;WEAVER DONALD;SUN SHENGGUO;MCLELLAN ALEXANDER;LU ERHU;
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申请日2016-08-05
分类号A61K31/045;A61K31/08;A61K31/194;A61K31/16;A61K31/131;A61K31/166;A61K31/11;A61K31/155;A61K31/10;A61K31/164;A61K31/18;A61K31/121;A61K31/133;A61K31/135;A61P25/04;A61P29;
国家 JP
入库时间 2022-08-21 14:02:05

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