Non-peptidyl, potent, and selective mu opioid receptor antagonists and their use in treating opioid addiction and opioid induced constipation

• 1. 吗啡与至少一种阿片拮抗剂的组合用于治疗阿片依赖性和用于防止阿片瘾患者非口服地滥用阿片制剂的用途 [P] . 中国专利： CN103893179A . 2014-07-02
• 2. 吗啡与至少一种阿片拮抗剂的组合用于治疗阿片依赖性和用于防止阿片瘾患者非口服地滥用阿片制剂的用途 [P] . 中国专利： CN101370503A . 2009-02-18
• 3. NON-PEPTIDYL, POTENT, AND SELECTIVE MU OPIOID RECEPTOR ANTAGONISTS AND THEIR USE IN TREATING OPIOID ADDICTION AND OPIOID INDUCED CONSTIPATION [P] . 美国专利： US2014371255A1 . 2014-12-18

  机译： 非肽，潜力和选择性MU阿片受体拮抗剂，及其在治疗阿片成瘾和阿片诱导性便秘中的用途

• 4. Non-peptidyl, potent, and selective mu opioid receptor antagonists [P] . 美国专利： US8772308B2 . 2014-07-08

  机译： 非肽基，有效和选择性的μ阿片受体拮抗剂

• 5. NON-PEPTIDYL, POTENT, AND SELECTIVE MU OPIOID RECEPTOR ANTAGONISTS [P] . 欧洲知识产权局专利： EP2387577A4 . 2012-10-17

  机译： 非肽，强效和选择性MU阿片受体拮抗剂

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