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Formulation comprising 1 h - quinazoline - 2, 4 - dione ampa receptor antagonists, in the form of immediate release tablets and preparation thereof
Formulation comprising 1 h - quinazoline - 2, 4 - dione ampa receptor antagonists, in the form of immediate release tablets and preparation thereof
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机译:速释片剂形式的包含1 h-喹唑啉-2,4-二酮安培受体拮抗剂的制剂及其制备
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摘要
Disclosed herein is a tablet comprising a hydroxypropylcellulose and an active ingredient selected from compounds of Formula (I) and salts thereof: wherein R1 represents CF3, CHF2, CH2F, CH3CHF-, CH3CF2-, ethyl or iso-propyl and R2 represents alkyl substituted by one or more substituents, the substituents being defined in the specification, and whereby the heterocycle is bound to the phenyl ring by a carbon-atom. Also disclosed is a process for preparing the above tablet. In one embodiment the compound it N-{ 6-[3-(1-hydroxy-ethyl)-phenyl]-2,4-dioxo-7-trifluoromethyl-1,4-dihydro-2H-quinazolin-3-yl} -methanesulfonamide.
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