Efficient synthesis of highly funetionalized Indoles and Indolines by C-H bond activation

机译：通过C-H键活化有效地合成高浊度吲哚和吲哚吲哚

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Direct oxidative C-C or C-heteroatom cross-coupling by selective C-H bond activation is a promising strategy for streamlining organic synthesis and, recently, many breakthroushs have been made. In our research, we want to facilitate the synthesis of important heterocvcles bv innovative C-H bond activation reactions. Consequently, we have developed new routes to indoles and mdolines, ubiquitous motifs of biologically active natural products: - a new synthesis of highly funetionalized indoles by direct C-H bond activation of substituted anilines (Figure 1a).

机译：通过选择性C-H键活化的直接氧化C-C或C-杂原子交叉偶联是精简有机合成的有希望的策略，最近已经进行了许多突破性。在我们的研究中，我们希望促进重要的杂交BV创新的C-H键活化反应的合成。因此，我们已经为吲哚和姆多洛尔开发了新的途径，无处不在的生物活性天然产品的主题： - 通过直接C-H键活化的取代苯胺的C-H键活化来新的高浊度吲哚（图1A）。

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《European Symposium on Organic Chemistry》|2009年||共1页
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T. Droge; J. J. Neumann; S. Rakshit;
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中图分类有机化学;
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1. Pd-catalyzed dehydrogenative C-H activation of iminyl hydrogen with the indole C3-H and C2-H bond: an elegant synthesis of indeno[1,2-b]indoles and indolo[1,2-a] indoles [J] . Hazra Somjit, Mondal Biplab, De Rajendra Narayan, RSC Advances . 2015,第29期

机译：Pd催化的吲哚C3-H和C2-H键亚氨基氢的C-H脱氢活化：吲哚[1,2-b]吲哚和吲哚[1,2-a]吲哚的精细合成
2. Merging C-H Activation and Alkene Difunctionalization at Room Temperature: A Palladium-Catalyzed Divergent Synthesis of Indoles and Indolines [J] . Manna Manash Kumar, Hossian Asik, Jana Ranjan Organic letters . 2015,第3期

机译：室温下合并C-H活化和烯烃双官能化：吲哚和吲哚的钯催化发散合成
3. Ruthenium(ii)-catalyzed selective C-H bond activation of imidamides and coupling with sulfoxonium ylides: an efficient approach for the synthesis of highly functional 3-ketoindoles [J] . Wu Chenglin, Zhou Jianhui, He Guoxue, Organic Chemistry Frontiers . 2019,第8期

机译：钌（II） - 催化咪酰胺的选择性C-H键活化和与亚磺氧化酰胺的偶联：合成高效3-酮吲哚的有效方法
4. Efficient synthesis of highly funetionalized Indoles and Indolines by C-H bond activation [C] . T. Droge, J. J. Neumann, S. Rakshit European Symposium on Organic Chemistry . 2009

机译：通过C-H键活化有效地合成高浊度吲哚和吲哚吲哚
5. Synthesis and Characterization of Group VIII & IX Transition Metal Complexes and Their Application in C-H Bond Activation and Hydrogen Transformation [D] . Yuan, Hongmei. 2018

机译：VIII和IX过渡金属配合物组的合成与表征及其在C-H键活化和氢转化中的应用
6. Fe(II)-Catalyzed Amination of Aromatic C-H Bonds via Ring Opening of 2H-Azirines: Synthesis of 23-Disubstituted Indoles [O] . Samaresh Jana, Mack D. Clements, Barry K. Sharp, -1

机译：的Fe（II） - 催化经由2H-azirines的开环芳族C-H键的胺化：23-二取代的吲哚的合成
7. Highly Efficient Copper-Catalyzed Nitro-Mannich Type Reaction: Cross-Dehydrogenative-Coupling between sp3 C-H Bond and sp3 C-H Bond [O] . -1

机译：高效铜催化的硝基 - 曼尼奇型反应：SP3 C-H键和SP3 C-H键之间的交叉脱氢偶联

Efficient synthesis of highly funetionalized Indoles and Indolines by C-H bond activation

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