Microwave Promoted Synthesis of Pharmacologically Active Pyrazolidinonyl Derivatives of Benzothiazoles

Krishnakant T Waghmode; Prachi K Shinde

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Microwave Promoted Synthesis of Pharmacologically Active Pyrazolidinonyl Derivatives of Benzothiazoles

机译：微波促进的苯并噻唑类药理活性吡唑二酮基衍生物的合成

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Microwave promoted synthesis of pharmacologically active N-(1,3-benzothiazol-2-yl)-2-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)amino]acetamides is described. Microwave assisted synthesis not only reduced the reaction time drastically but also gave excellent yields. The synthesized compounds are characterized by Fourier Transform Infra-Red (FTIR), Proton Nuclear Magnetic Resonance (1H-NMR) and mass spectral data.

机译：微波促进合成具有药理活性的N-（1,3-苯并噻唑-2-基）-2-[（1,5-二甲基-3-氧代-2-苯基-2,3-二氢-1H-吡唑-4-描述了（yl）氨基]乙酰胺。微波辅助合成不仅大大减少了反应时间，而且产率很高。合成的化合物的特征在于傅立叶变换红外（FTIR），质子核磁共振（1H-NMR）和质谱数据。

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《Der Pharma Chemica: journal for medicinal chemistry, pharmaceutical chemistry and computational chemistry》 |2017年第22期|共3页
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Krishnakant T Waghmode; Prachi K Shinde;
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Microwave Promoted Synthesis of Pharmacologically Active Pyrazolidinonyl Derivatives of Benzothiazoles

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