Efficient Microwave-Assisted Synthesis of Secondary Alkylpropargylamines by Using A3-Coupling with Primary Aliphatic Amines

Jitender B. Bariwal; Denis S. Ermolatev; Erik V. Van der Eycken

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Efficient Microwave-Assisted Synthesis of Secondary Alkylpropargylamines by Using A3-Coupling with Primary Aliphatic Amines

机译：A3-偶联初级脂肪胺的微波辅助高效合成仲烷基炔丙胺

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Multicomponent reactions (MCRs) have attracted much attention in the framework of combinatorial chemistry owing to their synthetic efficiency, intrinsic atom economy, high selectivity and procedural simplicity. These reactions constitute a valuable approach for the creation of large libraries of structurally related, drug-like compounds, thereby enabling rapid lead identification and optimisation in drug discovery. They represent environmentally friendly processes by reducing the number of steps, energy consumption and waste production.[1]

机译：多组分反应（MCR）的合成效率高，固有的原子经济性，高选择性和操作简便性，在组合化学领域引起了广泛关注。这些反应构成了创建大型结构相关的类药物化合物文库的有价值的方法，从而能够快速识别药物并优化药物发现。它们通过减少步骤数，减少能源消耗和减少废物产生来代表了环境友好型过程。[1]

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《Chemistry: A European journal》 |2010年第11期|共4页
作者
Jitender B. Bariwal; Denis S. Ermolatev; Erik V. Van der Eycken;
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正文语种 eng
中图分类应用化学;
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environmentally friendly; valuable approach; enabling rapid;

机译：环保;有价值的方法;快速实现;

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1. Efficient Microwave-Assisted Synthesis of Secondary Alkylpropargylamines by Using A3-Coupling with Primary Aliphatic Amines [J] . Jitender B. Bariwal, Denis S. Ermolatev, Erik V. Van der Eycken Chemistry: A European journal . 2010,第11期

机译：A3-偶联初级脂肪胺的微波辅助高效合成仲烷基炔丙胺
2. Terminal secondary C(sp3), aliphatic secondary C(sp2), aliphatic tertiary C(sp2), primary amine (aliphatic), ring secondary C(sp3) and imidazole numbers can be used to discriminate between cytokinins and cytokinin antagonists [J] . Andujar Ivan, Gomez Daviel, Perez Lianny, Plant Cell, Tissue and Organ Culture: An International Journal on in Vitro Culture of Higher Plants . 2019,第1期

机译：末端次级C（SP3），脂族次级C（SP2），脂族叔C（SP2），伯胺（脂族），环二次C（SP3）和咪唑数可用于区分细胞蛋白和细胞蛋白拮抗剂
3. THE USE OF BIS(AMINOL) ETHERS DERIVED FROM ALIPHATIC PRIMARY AMINES IN THE SYNTHESIS OF SECONDARY AND TERTIARY AMINES [J] . Heaney H., Papageorgiou G. Tetrahedron . 1996,第10期

机译：脂肪族初级胺衍生的双（氨基）醚在合成仲胺和叔胺中的应用
4. DERIVATIZATION-FREE ANALYSIS OF VOLATILE ALIPHATIC AND AROMATIC PRIMARY, SECONDARY AND TERTIARY AMINES IN INDOOR AIR BY HPLC-ESI-MS [C] . M Rampfl, F Mayer, K Breuer, Indoor Air 2005 . 2005

机译：高效液相色谱-ESI-MS分析室内空气中的挥发性脂族和芳族主要，二次和叔胺
5. Part A. Diastereoselective synthesis of protected secondary amines via reduction /alkylation or deprotonation /alkylation of N-diphenylphosphinylimines. Part B. Synthesis of secondary amines via 1,2-addition of organometallic reagents to N-diphenylphosphinylimines and subsequent alkylation [D] . Shin, Hyunshun 2001

机译：A部分：通过N-二苯基膦亚胺的还原/烷基化或去质子化/烷基化的非对映选择性合成保护的仲胺。 B部分：通过将有机金属试剂1,2-加成到N-二苯基膦亚胺和随后的烷基化反应来合成仲胺
6. Efficient microwave-assisted synthesis of amine substituted pentafluorophenylporphyrin [O] . Diana Samaroo, Clifford E. Soll, Louis J. Todaro, -1

机译：微波辅助合成胺取代的五氟苯基卟啉
7. Synthesis of Some Novel α-Cyanoketene-N,S-acetals Derived from Secondary Aliphatic Amines and Their Use in Pyrazole Synthesis [O] . Wedad M. Al-Adiwish, M. I. M. Tahir, W. A. Yaacob 2013

机译：一些新型α-氰基乙烯-N，S-缩醛的合成及其在吡唑合成中的应用
8. Alkylation of Amines: A New Method for the Synthesis of Quaternary Ammonium Compounds from Primary and Secondary Amines [R] . Sommer, H. Z., Jackson, L. L. 1969

机译：胺的烷基化：从伯胺和仲胺合成季铵化合物的新方法

Efficient Microwave-Assisted Synthesis of Secondary Alkylpropargylamines by Using A3-Coupling with Primary Aliphatic Amines

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