Synthesis and antimicrobial screening of novel bis-triazolo-dithiadiazines containing bridgehead nitrogen

Deohate Pradip P.; Kawle Pravin R.

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Synthesis and antimicrobial screening of novel bis-triazolo-dithiadiazines containing bridgehead nitrogen

机译：新型含桥头氮的双-三唑并二硫杂二嗪的合成与抗菌筛选

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1,4-Bis-(3-arylimino-[1,2,4]-triazolo-[3,4-c]-[1,2,4,5]-dithiadiazin-6-yl)-benzenes have been synthesized by treating 1,4-bis-(4-amino-3-mercapto-4H[1,2,4]-triazol-5-yl-benzene with N-aryl-S-chloro isothiocarbamoyl chlorides and then basification with dilute ammonia solution. Synthesis of 1,4-bis-(4-amino-3-mercapto-4H-[1,2,4]-triazol-5-yl-benzene was carried out by interacting the terephthalic acid dihydrazide with carbondisulphide in presence of potassium hydroxide and then by adding the hydrazine hydrate. Bis-triazolo-dithiadiazines on acetylation afforded di-acetyl derivatives. Structures of title compounds were delineated on the basis of determination of equivalent weight, chemical transformation, elemental analysis and spectral studies. These compounds have been assayed for their antibacterial and antifungal activity against various micro-organisms.

机译：合成了1,4-双-（3-芳基-[1,2,4]-三唑-[3,4-c]-[1,2,4,5]-二噻二嗪-6-基）-苯用N-芳基-S-氯异硫代氨基甲酰氯处理1,4-双-（4-氨基-3-巯基-4H [1,2,4]-三唑-5-基苯，然后用稀氨水碱化通过在钾的存在下使对苯二甲酸二酰肼与二硫化碳相互作用来合成1,4-双-（4-氨基-3-巯基-4H- [1,2,4]-三唑-5-基苯氢氧化物然后加入水合肼，双-三唑并二硫代二嗪经乙酰化得到二乙酰基衍生物，在确定当量，化学转化，元素分析和光谱研究的基础上勾勒出标题化合物的结构。分析它们对各种微生物的抗菌和抗真菌活性。

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《Journal of the Indian Chemical Society》 |2015年第6期|共4页
作者
Deohate Pradip P.; Kawle Pravin R.;
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正文语种 eng
中图分类化学;
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Novel bis-triazolo-dithiadiazines; synthesis; antimicrobial activity;

机译：新型双三唑并二硫杂二嗪;合成;抗菌活性;

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1. Synthesis and antimicrobial screening of novel bis-triazolo-dithiadiazines containing bridgehead nitrogen [J] . Deohate Pradip P., Kawle Pravin R. Journal of the Indian Chemical Society . 2015,第6期

机译：新型含桥头氮的双-三唑并二硫杂二嗪的合成与抗菌筛选
2. Synthesis, structural study and antimicrobial screening of bridgehead nitrogen containing 1,8-bis-thiadiazino-triazolyl-octanes [J] . Rajesh M. Kharate, Pradip P. Deohate, B. N. Berad Der Pharma Chemica: journal for medicinal chemistry, pharmaceutical chemistry and computational chemistry . 2012,第6期

机译：含1,8-双-噻二氮杂-三唑基辛烷的桥头含氮化合物的合成，结构研究和抗菌筛选
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机译：缩合桥头氮杂环系统：噻唑[3'，2'：2，3]-三嗪[5，6-b]吲哚和异构体噻唑[2'，3'：3，4]-的合成及抑菌活性as-triazino [5，6-b]吲哚8。8的明确合成也有蜜蜂
4. Biosynthesis, characterization of silver nanoparticles and antimicrobial screening by Oscillatoria Annae [C] . S. Geetha, K. Vijayakumar, K. R. Aranganayagam, International Conference on Physics and Chemistry of Materials in Novel Engineering Applications . 2020

机译：生物合成，银纳米粒子的表征和振荡器Annae的抗微生物筛选
5. THE EFFECTS OF CARBADOX, A SYNTHETIC ANTIMICROBIAL AGENT, ON GROWTH, NITROGEN BALANCE, PROTEIN SYNTHESIS, PROTEIN DEGRADATION AND APPARENT AMINO ACID ABSORPTION IN THE GROWING PIG [D] . BAJJALIEH, NICHOLI LLOYD 1980

机译：合成抗微生物剂碳水化合物对生长猪生长，氮平衡，蛋白质合成，蛋白质降解和表观氨基酸吸收的影响
6. Synthesis Biological Evaluation and ComputationalStudies of Tri- and Tetracyclic Nitrogen-Bridgehead Compounds as PotentDual-Acting AChE Inhibitors and hH3 ReceptorAntagonists [O] . Fouad H. Darras, Steffen Pockes, Guozheng Huang, 2014

机译：合成生物学评估和计算三环和四环氮桥头化合物的研究双作用AChE抑制剂和hH3受体拮抗剂
7. Heterocyclic systems containing bridgehead nitrogen atom: Synthesis and antimicrobial activity of thiadiazolo2′,3′:2,3imidazo4,5-Bquinoxaline [O] . Teja Ramakrishna, Kapu Sivakrishna, Kadiyala Swapana, 2016

机译：含桥头氮原子的杂环系统：噻二唑2'，3'：2,3咪唑4,5-B喹喔啉的合成及抑菌活性
8. Synthesis of Bridgehead Nitrogen Heterocycles [R] . Scovill, J. P., Burckhalter, J. H. 1979

机译：桥头氮杂环化合物的合成

Synthesis and antimicrobial screening of novel bis-triazolo-dithiadiazines containing bridgehead nitrogen

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