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ANTICANCER COMBINATION OF ARTEMISININ-BASED DRUGS AND OTHER CHEMOTHERAPEUTIC AGENTS

机译:青蒿素类药物和其他化学治疗剂的抗癌药组合

摘要

THE PRESENT INVENTION RELATES TO COMBINATIONS BETWEEN ARTEMISININ-BASED POTENT ANTI-MALARIAL AGENTS, SELECTED FROM THE GROUP CONSISTING OF ART, DHA AND ARM, AND A FURTHER CHEMOTHERAPEUTIC DRUG SELECTED FROM THE GROUP CONSISTING OF A CAMPTOTHECIN DERIVATIVE, OR A PARP-1 INHIBITOR, OR AN INTERCALATING DNA AGENT, OR AN ALKYLATING AGENT. SUCH COMBINATIONS, SHOWED MEDIUM TO STRONG SYNERGISM IN VARIOUS MODELS OF CANCER, IN PARTICULAR IN NSCL.
机译:本发明涉及选自由ART,DHA和ARM组成的组的基于青蒿素的潜在抗疟疾剂的组合,以及选自由喜树碱衍生物,或PARP-1抑制剂组成的组的进一步化疗药物的组合。或可插入的DNA代理或烷基化代理。在NSCL的各种模型中,将这种组合显示为中等至强的协同效应。

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