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ANTICANCER COMBINATION OF ARTEMISININ-BASED DRUGS AND OTHER CHEMOTHERAPEUTIC AGENTS
ANTICANCER COMBINATION OF ARTEMISININ-BASED DRUGS AND OTHER CHEMOTHERAPEUTIC AGENTS
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机译:青蒿素类药物和其他化学治疗剂的抗癌药组合
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摘要
THE PRESENT INVENTION RELATES TO COMBINATIONS BETWEEN ARTEMISININ-BASED POTENT ANTI-MALARIAL AGENTS, SELECTED FROM THE GROUP CONSISTING OF ART, DHA AND ARM, AND A FURTHER CHEMOTHERAPEUTIC DRUG SELECTED FROM THE GROUP CONSISTING OF A CAMPTOTHECIN DERIVATIVE, OR A PARP-1 INHIBITOR, OR AN INTERCALATING DNA AGENT, OR AN ALKYLATING AGENT. SUCH COMBINATIONS, SHOWED MEDIUM TO STRONG SYNERGISM IN VARIOUS MODELS OF CANCER, IN PARTICULAR IN NSCL.
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