Synthesis and Biological Activity of N-Aryl-Na??-Heteroaryl Carbamides

S. N. P; eya; Vaishali Mishra; Alka P

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Synthesis and Biological Activity of N-Aryl-Na??-Heteroaryl Carbamides

机译：N-芳基-Na +-杂芳基碳酰胺的合成及生物活性

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A series of N-aryl-N’-heteroaryl carbamides were synthesized. The structure of the compounds was established by means of I. R., 1HNMR, Mass spectra and elemental analysis. All the compounds were screened for their antibacterial and antifungal activities. Compound 3e with chlorosubstitution was most active as antibacterial and antifungal with MIC of 0.075 mg/mL against E. coli and P. aruginosa.

机译：合成了一系列的N-芳基-N’-杂芳基脲。通过IR，1 HNMR，质谱和元素分析确定化合物的结构。筛选所有化合物的抗菌和抗真菌活性。具有氯取代作用的化合物3e作为抗菌和抗真菌活性最高，对大肠杆菌和古铜假单胞菌的MIC为0.075 mg / mL。

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《Der Pharma Chemica: journal for medicinal chemistry, pharmaceutical chemistry and computational chemistry》 |2010年第3期|共7页
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S. N. P; eya; Vaishali Mishra; Alka P;
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Synthesis and Biological Activity of N-Aryl-Na??-Heteroaryl Carbamides

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