机译:Discovery of a Novel Class of PROTACs as Potent and Selective Estrogen Receptor alpha Degraders to Overcome Endocrine-Resistant Breast Cancer In Vitro and In Vivo
机译:Design, Synthesis, and Evaluation of (R)-8-((Tetrahydrofuran-2-yl)methyl)pyrido2,3-dpyrimidin-7-ones as Novel Selective ACK1 Inhibitors to Combat Acquired Resistance to the Third-Generation EGFR Inhibitor
机译:psi and chi Angle Constrains at the C-Terminus Trp Position of the Melanotropin Tetrapeptide Ac-His-D-Phe-Arg-Trp-NH2 Lead to Potent and Selective Agonists at hMC1R and hMC4R
机译:Prodrug Strategies for the Development of beta-L-5-((E)-2-Bromovinyl)-1-((2S,4S)-2-(hydroxymethyl)-1,3-(dioxolane-4-yl))uracil (L-BHDU) against Varicella Zoster Virus (VZV)
机译:X-ray Crystal Structure-Guided Discovery of Novel Indole Analogues as Colchicine-Binding Site Tubulin Inhibitors with Immun Potentiating and Antitumor Effects against Melanoma
机译:Discovery of Nanomolar Melanocortin-3 Receptor (MC3R)-Selective Small Molecule Pyrrolidine Bis-Cyclic Guanidine Agonist Compounds Via a High Throughput 'Unbiased' Screening Campaign (vol 64, pg 5577, 2021)