Arylsulfonyl acridinyl derivatives acting on Plasmodium falciparum.

Santelli Rouvier C; Pradines B; Berthelot M; Parzy D; Barbe J

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Arylsulfonyl acridinyl derivatives acting on Plasmodium falciparum.

机译：作用于恶性疟原虫的芳基磺酰基a啶基衍生物。

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Several arylacridinyl sulfones have been synthesized and their antimalarial action was tested on Plasmodium falciparum. PABA (para-aminobenzoic acid) has no antagonistic effect with these compounds as opposed to the observed effect with dapsone and sulfonamides previously studied. A possible relationship between the ability of cleavage of the S-9C acridinic bond and activity is suggested.

机译：已经合成了几种芳基吡啶基砜，并在恶性疟原虫上测试了它们的抗疟作用。与先前研究的氨苯砜和磺酰胺类药物相比，PABA（对氨基苯甲酸）对这些化合物没有拮抗作用。建议S-9C C啶键的裂解能力与活性之间可能存在关系。

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《European Journal of Medicinal Chemistry: Chimie Therapeutique》 |2004年第9期|共10页
作者
Santelli Rouvier C; Pradines B; Berthelot M; Parzy D; Barbe J;
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正文语种 eng
中图分类基础医学;
关键词
Plasmodium falciparum; derivatives; 4-Aminobenzoic Acid; Dapsone; 疟原虫; 恶性; 4-氨基苯甲酸; 氨苯砜;

机译：Plasmodium falciparum;derivatives;4-Aminobenzoic Acid;Dapsone;疟原虫;恶性;4-氨基苯甲酸;氨苯砜;

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1. Arylsulfonyl acridinyl derivatives acting on Plasmodium falciparum. [J] . Santelli Rouvier C, Pradines B, Berthelot M, European Journal of Medicinal Chemistry: Chimie Therapeutique . 2004,第9期

机译：作用于恶性疟原虫的芳基磺酰基a啶基衍生物。
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Arylsulfonyl acridinyl derivatives acting on Plasmodium falciparum.

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