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机译:N-萘甲酰对纳曲胺(NNTA),μ/κ阿片类异构体的高度选择性和有效活化剂
Department of Medicinal Chemistry, College of Pharmacy, University of Minnesota, Minneapolis, MN 55455,Department of Pharmacology,University of Minnesota, Minneapolis, MN 55455;
Department of Medicinal Chemistry, College of Pharmacy, University of Minnesota, Minneapolis, MN 55455;
Department of Medicinal Chemistry, College of Pharmacy, University of Minnesota, Minneapolis, MN 55455;
Department of Medicinal Chemistry, College of Pharmacy, University of Minnesota, Minneapolis, MN 55455;
Department of Neuroscience, Medical School, University of Minnesota, Minneapolis, MN 55455;
Department of Pharmacology, Toxicology, and Neuroscience, Louisiana State University Health Science Center,Shreveport, LA 71115;
Department of Medicinal Chemistry, College of Pharmacy, University of Minnesota, Minneapolis, MN 55455,Department of Pharmacology,University of Minnesota, Minneapolis, MN 55455,Department of Neuroscience, Medical School, University of Minnesota, Minneapolis, MN 55455;
机译:新型TIPP(H-Tyr-Tic-Phe-Phe-OH)类似物在δ阿片受体上显示出广泛的功效。发现了两种高效和选择性的δ阿片激动剂
机译:两种新的阿片类药物δ受体配体:体外分离制剂中的高选择性激动剂和有效选择性拮抗剂。
机译:作为高度选择性神经肽FF1受体拮抗剂的鉴定N-酰化 - (d)arg-leu-NH2二肽,其致力于防止阿片类药物诱导的痛觉
机译:具有高效激动剂和拮抗剂/激动剂阿片类能活性DMT-TIC类似物的合成与药理活性
机译:合成Salvinorin支架以开发潜在的止痛药和选择性,有效的阿片样物质配体
机译:N-萘甲酰-β-纳曲胺(NNTA)μ/κ阿片类异构体的高度选择性和有效活化剂
机译:N-萘甲酰-β-纳曲胺(NNTA),μ/κ阿片类异构体的高度选择性和有效活化剂